日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

In Vitro and In Silico Biological Studies of 4-Phenyl-2-quinolone (4-PQ) Derivatives as Anticancer Agents

4-苯基-2-喹诺酮(4-PQ)衍生物作为抗癌剂的体外和计算机生物学研究

Chen, Yi-Fong; Lawal, Bashir; Huang, Li-Jiau; Kuo, Sheng-Chu; Sumitra, Maryam Rachmawati; Mokgautsi, Ntlotlang; Lin, Hung-Yun; Huang, Hsu-Shan

Synthesis and antitumor activity of bis(hydroxymethyl)propionate analogs of pterostilbene in cisplatin-resistant human oral cancer cells

紫檀芪双(羟甲基)丙酸酯类似物在顺铂耐药人口腔癌细胞中的合成及抗肿瘤活性

Hsieh, Min-Tsang; Huang, Li-Jiau; Wu, Tian-Shung; Lin, Hui-Yi; Morris-Natschke, Susan L; Lee, Kuo-Hsiung; Kuo, Sheng-Chu

α-Carboline derivative TJY-16 inhibits tumor growth by inducing G2/M cell cycle arrest in glioma cells

α-咔啉衍生物TJY-16通过诱导胶质瘤细胞G2/M期细胞周期阻滞来抑制肿瘤生长。

Huang, Hsiao-Chieh; Liu, Wei-Ting; Hua, Kuo-Su; Hung, Hui-Chi; Tsai, Jui-Ying; Kuo, Sheng-Chu; Huang, Li-Jiau; Gean, Po-Wu

Design and synthesis of new 2-arylnaphthyridin-4-ones as potent antitumor agents targeting tumorigenic cell lines

设计和合成新型 2-芳基萘啶-4-酮作为针对致瘤细胞系的有效抗肿瘤药物

Chin-Yu Liu, Yung-Yi Cheng, Ling-Chu Chang, Li-Jiau Huang, Li-Chen Chou, Chi-Hung Huang, Meng-Tung Tsai, Chih-Chang Liao, Mei-Hua Hsu, Hui-Yi Lin, Tian-Shung Wu, Yen-Fang Wen, Yu Zhao, Sheng-Chu Kuo, Kuo-Hsiung Lee

BC3EE2,9B, a synthetic carbazole derivative, upregulates autophagy and synergistically sensitizes human GBM8901 glioblastoma cells to temozolomide

BC3EE2,9B 是一种合成咔唑衍生物,可上调自噬并协同增强人类 GBM8901 胶质母细胞瘤细胞对替莫唑胺的敏感性

Chien-Min Chen, Jhih-Pu Syu, Tzong-Der Way, Li-Jiau Huang, Sheng-Chu Kuo, Chung-Tien Lin, Chih-Li Lin

YC-1 inhibits proliferation of breast cancer cells by down-regulating EZH2 expression via activation of c-Cbl and ERK

YC-1通过激活c-Cbl和ERK下调EZH2表达来抑制乳腺癌细胞增殖

Ling-Chu Chang, Hui-Yi Lin, Meng-Tung Tsai, Ruey-Hwang Chou, Fang-Yu Lee, Che-Ming Teng, Min-Tsang Hsieh, Hsin-Yi Hung, Li-Jiau Huang, Yung-Luen Yu, Sheng-Chu Kuo

Three new clerodane diterpenes from Polyalthia longifolia var. pendula

从垂枝暗罗(Polyalthia longifolia var. pendula)中分离得到三种新的克罗丹二萜类化合物。

Wu, Tung-Ho; Cheng, Yung-Yi; Chen, Chao-Jung; Ng, Lean-Teik; Chou, Li-Chen; Huang, Li-Jiau; Chen, Yung-Husan; Kuo, Sheng-Chu; El-Shazly, Mohamed; Wu, Yang-Chang; Chang, Fang-Rong; Liaw, Chih-Chuang

Design, synthesis, and mechanism of action of 2-(3-hydroxy-5-methoxyphenyl)-6-pyrrolidinylquinolin-4-one as a potent anticancer lead

2-(3-羟基-5-甲氧基苯基)-6-吡咯烷基喹啉-4-酮作为一种强效抗癌先导化合物的设计、合成及作用机制研究

Cheng, Yung-Yi; Liu, Chin-Yu; Tsai, Meng-Tung; Lin, Hui-Yi; Yang, Jai-Sing; Wu, Tian-Shung; Kuo, Sheng-Chu; Huang, Li-Jiau; Lee, Kuo-Hsiung

Synthesis and cytotoxicity of 1,6,8,9-substituted α-carboline derivatives

1,6,8,9-取代α-咔啉衍生物的合成及细胞毒性

Tsai, Jui-Ying; Lin, Yi-Chien; Hsu, Mei-Hua; Kuo, Sheng-Chu; Huang, Li-Jiau

The anti-inflammatory carbazole, LCY-2-CHO, inhibits lipopolysaccharide-induced inflammatory mediator expression through inhibition of the p38 mitogen-activated protein kinase signaling pathway in macrophages

抗炎咔唑 LCY-2-CHO 通过抑制巨噬细胞中的 p38 丝裂原活化蛋白激酶信号通路来抑制脂多糖诱导的炎症介质表达

Feng-Ming Ho, Chih-Chang Lai, Li-Jiau Huang, Tsun Cheng Kuo, Chien M Chao, Wan-Wan Lin