日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Long-acting GIPR agonist LY3537021 reduces body weight and fasting blood glucose in patients with T2D: Preclinical development and phase 1 randomized ascending dose studies

长效GIPR激动剂LY3537021可降低2型糖尿病患者的体重和空腹血糖:临床前开发和1期随机递增剂量研究

Roell, William; Alsina-Fernandez, Jorge; Qu, Hongchang; Coskun, Tamer; Benson, Charles; Haupt, Axel; Kelly, Ronan P; O'Farrell, Libbey; Sloop, Kyle W; Steele, James P; Ficorilli, James; Regmi, Ajit; Rettiganti, Mallikarjuna; Urva, Shweta; Mather, Kieren J; Pratt, Edward

GLP-1R biased cAMP agonism maintains glycemic control with reduced malaise and emesis in preclinical mammalian models

在临床前哺乳动物模型中,GLP-1R 偏向性 cAMP 激动剂作用可维持血糖控制,并减少不适和呕吐。

Baumer-Harrison, Caitlin; Aldaghma, Danya; White, Alex D; Applebey, Sarah V; Pataro, Allison M; Mohiby, Allaha Z; Alonso, Brandon; Xiao, Allison G; O'Farrell, Libbey S; Qian, Yuewei; Coskun, Tamer; Coghlan, Matthew P; Willard, Francis S; Ai, Minrong; Sloop, Kyle W; Doyle, Robert P; Borner, Tito; De Jonghe, Bart C; Hayes, Matthew R

Eloralintide (LY3841136), a novel amylin receptor agonist for the treatment of obesity: From discovery to clinical proof of concept

埃洛拉林肽(LY3841136),一种用于治疗肥胖症的新型胰淀素受体激动剂:从发现到临床概念验证

Briere, Daniel A; Qu, Hongchang; Lansu, Katherine; He, Minxia Michelle; Moyers, Julie S; Coskun, Tamer; Long, Annie; Allen, Dawn; O'Farrell, Libbey; Bowen, Breanna; Pratt, Edward; Tidemann-Miller, Beth; Tham, Lai San; Ibriga, Hilda; Alsina-Fernandez, Jorge; Mather, Kieren J; Haupt, Axel; Bhattachar, Shobha N

Characterization of LY3324954 a long-acting glucagon-receptor agonist

LY3324954(一种长效胰高血糖素受体激动剂)的特性分析

Roell, William; Coskun, Tamer; Kim, Teayoun; O'Farrell, Libbey; Martin, Jennifer A; Nason, Shelly; Hernandez-Alamillo, Jasmin; Dhantu, Saidharshana; Drucker, Daniel J; Sloop, Kyle W; Steele, James P; Alsina-Fernandez, Jorge; Habegger, Kirk M

GIPR Agonism Enhances TZD-Induced Insulin Sensitivity in Obese IR Mice

GIPR 激动剂增强肥胖 IR 小鼠中 TZD 诱导的胰岛素敏感性

Ellen C Furber, Karissa Hyatt, Kyla Collins, Xinxin Yu, Brian A Droz, Adrienne Holland, Jessica L Friedrich, Samantha Wojnicki, Debra L Konkol, Libbey S O'Farrell, Hana E Baker, Tamer Coskun, Philipp E Scherer, Christine M Kusminski, Michael E Christe, Kyle W Sloop, Ricardo J Samms

Glutamate Transport Proteins and Metabolic Enzymes are Poor Prognostic Factors in Invasive Lobular Carcinoma

谷氨酸转运蛋白和代谢酶是侵袭性小叶癌的不良预后因素

Todd A Young, Shaymaa Bahnassy, Theresa C Abalum, Eden A Pope, Amanda Torres Rivera, Aileen I Fernandez, Ayodeji O Olukoya, Dua Mobin, Suman Ranjit, Nicole E Libbey, Sonali Persaud, Aaron M Rozeboom, Krysta Chaldekas, Brent T Harris, Zeynep Madak-Erdogan, Joseph L Sottnik, Matthew J Sikora, Rebecca

Morbillivirus: A highly adaptable viral genus

麻疹病毒属:一个适应性极强的病毒属

Libbey, Jane E; Fujinami, Robert S

Study protocol: Type III hybrid effectiveness-implementation study implementing Age-Friendly evidence-based practices in the VA to improve outcomes in older adults

研究方案:一项III型混合效果-实施研究,旨在评估在退伍军人事务部实施老年友好型循证实践以改善老年人预后的效果。

Piazza, Kirstin Manges; Ashcraft, Laura Ellen; Rose, Liam; Hall, Daniel E; Brown, Rebecca T; Bowen, Mary Elizabeth Libbey; Mavandadi, Shahrzad; Brecher, Alison C; Keddem, Shimrit; Kiosian, Bruce; Long, Judith A; Werner, Rachel M; Burke, Robert E

Microbial Characterization, Factors Contributing to Contamination, and Household Use of Cistern Water, U.S. Virgin Islands

美属维尔京群岛蓄水池水的微生物特征、污染因素及家庭用水情况

Rao, Gouthami; Kahler, Amy; Voth-Gaeddert, Lee E; Cranford, Hannah; Libbey, Stephen; Galloway, Renee; Molinari, Noelle-Angelique; Ellis, Esther M; Yoder, Jonathan S; Mattioli, Mia C; Ellis, Brett R

GIPR agonism mediates weight-independent insulin sensitization by tirzepatide in obese mice

GIPR 激动剂介导肥胖小鼠体重不依赖的胰岛素增敏作用

Ricardo J Samms, Michael E Christe, Kyla Al Collins, Valentina Pirro, Brian A Droz, Adrienne K Holland, Jessica L Friedrich, Samantha Wojnicki, Debra L Konkol, Richard Cosgrove, Ellen Ps Conceição Furber, Xiaoping Ruan, Libbey S O'Farrell, Annie M Long, Mridula Dogra, Jill A Willency, Yanzhu Lin, Li