日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Rapid and long-lasting antidepressant-like effects of the pituitary adenylate cyclase-activating polypeptide receptor antagonist PA-915 in chronic stress mouse models

垂体腺苷酸环化酶激活多肽受体拮抗剂PA-915在慢性应激小鼠模型中表现出快速且持久的抗抑郁样作用

Shintani, Yusuke; Hayata-Takano, Atsuko; Takasaki, Ichiro; Kurihara, Takashi; Miyata, Atsuro; Yamano, Yui; Ikuta, Manato; Takeshita, Rei; Murata, Kenichiro; Oguri, Taisei; Asaka, Chiaki; Nunomura, Kazuto; Lin, Bangzhong; Nakagawa, Shinsaku; Okada, Takuya; Toyooka, Naoki; Takumi, Toru; Ago, Yukio; Takuma, Kazuhiro; Hashimoto, Hitoshi

Compound Library Screening Identified Cladribine as a Novel Radiosensitizer for Prostate Cancer

化合物库筛选发现克拉屈滨是一种新型前列腺癌放射增敏剂

Oka, Toshiki; Hatano, Koji; Katsuki, Shohei; Kanaki, Tomohiro; Inoguchi, Shunsuke; Tani, Masaru; Yoshimura, Akihiro; Horibe, Yuki; Liu, Yutong; Sassi, Nesrine; Okuda, Yohei; Yamamoto, Akinaru; Uemura, Toshihiro; Yamamichi, Gaku; Ishizuya, Yu; Hayashi, Takuji; Yamamoto, Yoshiyuki; Kato, Taigo; Kawashima, Atsunari; Tamari, Keisuke; Lin, Bangzhong; Tani, Akiyoshi; Tsujikawa, Kazutake; Takahashi, Yutaka; Ogawa, Kazuhiko; Lupold, Shawn E; Nonomura, Norio

Discovery of a Selective Inhibitor of ZIP14 with Therapeutic Potential for Cancer-associated Cachexia

发现一种具有治疗癌症相关恶病质潜力的ZIP14选择性抑制剂

Hara, Takafumi; Tanaka, Gen; Tamura, Tomonori; Terajima, Masaomi; Hamamura, Kengo; Yoshida, Yuya; Kimura, Toru; Kasai, Yusuke; Nakayama, Yuta; Umeyama, Takumi; Hosoi, Kohei; Noguchi, Ayaka; Nakai, Yasuno; Hijikata, Atsushi; Matsukawa, Koji; Ujihara, Satoru; Kawabe, Tetsuhiro; Taguchi, Hiroki; Fujishiro, Hitomi; Jenkitkasemwong, Supak; Nunomura, Kazuto; Lin, Bangzhong; Fukunaka, Ayako; Yoshigai, Emi; Mishima, Kenji; Nakagawa, Shinsaku; Knutson, Michell D; Imagawa, Hiroshi; Matsunaga, Naoya; Ohdo, Shigehiro; Hamachi, Itaru; Sakurai, Hiroyuki; Fukada, Toshiyuki

Development of a high-throughput screening system targeting the protein-protein interactions between PRL and CNNM.

开发针对PRL和CNNM之间蛋白质-蛋白质相互作用的高通量筛选系统

Funato Yosuke, Mimura Mai, Nunomura Kazuto, Lin Bangzhong, Fujii Shintarou, Haruta Junichi, Miki Hiroaki

Anti-Schistosomal activity and ADMET properties of 1,2,5-oxadiazinane-containing compound synthesized by visible-light photoredox catalysis

可见光光氧化还原催化合成的含1,2,5-噁二嗪烷化合物的抗血吸虫活性和ADMET性质

Itoh, Kennosuke; Nakahara, Hiroki; Takashino, Atsushi; Hara, Aya; Katsuno, Akiho; Abe, Yuriko; Mizuguchi, Takaaki; Karaki, Fumika; Hirayama, Shigeto; Nagai, Kenichiro; Seki, Reiko; Sato, Noriko; Okuyama, Kazuki; Hashimoto, Masashi; Tokunaga, Ken; Ishida, Hitoshi; Mikami, Fusako; Kwofie, Kofi Dadzie; Kawada, Hayato; Lin, Bangzhong; Nunomura, Kazuto; Kanai, Toshio; Hatta, Takeshi; Tsuji, Naotoshi; Haruta, Junichi; Fujii, Hideaki

Design, Synthesis, and Monoamine Oxidase B Selective Inhibitory Activity of N-Arylated Heliamine Analogues

N-芳基化海拉明类似物的设计、合成及其对单胺氧化酶B的选择性抑制活性

Yamada, Makito; Hirose, Yu; Lin, Bangzhong; Fumimoto, Megumi; Nunomura, Kazuto; Natchanun, Sirimangkalakitti; Takahashi, Naoyuki; Ohki, Yuuta; Sako, Makoto; Murai, Kenichi; Harada, Kazuo; Arai, Masayoshi; Suzuki, Sayo; Nakamura, Tomonori; Haruta, Junichi; Arisawa, Mitsuhiro

Discovery of Benzylpiperazine Derivatives as CNS-Penetrant and Selective Histone Deacetylase 6 Inhibitors

发现苄基哌嗪衍生物作为中枢神经系统穿透性和选择性组蛋白去乙酰化酶6抑制剂

Hashimoto, Kosuke; Ide, Soichiro; Arata, Mayumi; Nakata, Akiko; Ito, Akihiro; Ito, Takashi K; Kudo, Norio; Lin, Bangzhong; Nunomura, Kazuto; Tsuganezawa, Keiko; Yoshida, Minoru; Nagaoka, Yasuo; Sumiyoshi, Takaaki

A novel RyR1-selective inhibitor prevents and rescues sudden death in mouse models of malignant hyperthermia and heat stroke

一种新型的RyR1选择性抑制剂能够预防和挽救恶性高热和中暑小鼠模型中的猝死

Yamazawa, Toshiko; Kobayashi, Takuya; Kurebayashi, Nagomi; Konishi, Masato; Noguchi, Satoru; Inoue, Takayoshi; Inoue, Yukiko U; Nishino, Ichizo; Mori, Shuichi; Iinuma, Hiroto; Manaka, Noriaki; Kagechika, Hiroyuki; Uryash, Arkady; Adams, Jose; Lopez, Jose R; Liu, Xiaochen; Diggle, Christine; Allen, Paul D; Kakizawa, Sho; Ikeda, Keigo; Lin, Bangzhong; Ikemi, Yui; Nunomura, Kazuto; Nakagawa, Shinsaku; Sakurai, Takashi; Murayama, Takashi

Discovery of peroxisome proliferator-activated receptor α (PPARα) activators with a ligand-screening system using a human PPARα-expressing cell line

利用人PPARα表达细胞系的配体筛选系统发现过氧化物酶体增殖物激活受体α (PPARα) 激活剂

Tachibana, Keisuke; Yuzuriha, Tomohiro; Tabata, Ryotaro; Fukuda, Syohei; Maegawa, Takashi; Takahashi, Rika; Tanimoto, Keiichi; Tsujino, Hirofumi; Nunomura, Kazuto; Lin, Bangzhong; Matsuura, Yoshiharu; Tanaka, Toshiya; Hamakubo, Takao; Sakai, Juro; Kodama, Tatsuhiko; Kobayashi, Tadayuki; Ishimoto, Kenji; Miyachi, Hiroyuki; Doi, Takefumi