日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Discovery of Covalent Ligands with AlphaFold3

利用 AlphaFold3 发现共价配体

Shamir, Yoav; Gabizon, Ronen; Rogel, Adi; Lin, David Yin-Wei; Andreotti, Amy H; London, Nir

Modulating the Binding Kinetics of Bruton's Tyrosine Kinase Inhibitors through Transition-State Effects

通过过渡态效应调节布鲁顿酪氨酸激酶抑制剂的结合动力学

Bravo, Eduardo Jr; Li, Yong; Lin, David Yin-Wei; Srinivasan, Bharath; Barone, Marco; Li, Stan Xiaogang; DelloRusso, Francesca; Rahiyanath, Anza Suneer; Corrionero, Ana; Alfonso, Patricia; Prendiville, Niall; Kozakov, Dima; Andreotti, Amy H; Tonge, Peter J

Screening and Characterization of Allosteric Small Molecules Targeting Bruton's Tyrosine Kinase.

筛选和表征靶向布鲁顿酪氨酸激酶的变构小分子

Kueffer Lauren E, Lin David Yin-Wei, Amatya Neha, Serrenho Joseph, Joseph Raji E, Courtney Adam H, Andreotti Amy H