日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Yeast Display Technology Enables Rapid Discovery of Low-Nanomolar Macrocyclic Peptide Inhibitors of Human Angiotensin-Converting Enzyme 2

酵母展示技术可快速发现低纳摩尔级人血管紧张素转化酶2大环肽抑制剂

Romanyuk, Zhanna; Bettin, Giacomo; Brear, Paul; Linciano, Sara; Mazzocato, Ylenia; Bonadies, Simone; Zanotto, Ilaria; Mazzucco, Camilla; Monferone, Alan; Soler, Miguel A; Pasut, Gianfranco; Martin, Sara De; Scarso, Alessandro; Heinis, Christian; Rothenberger, Sylvia; Hyvönen, Marko; Angelini, Alessandro

Targeting Autoinducer‑2 Quorum Sensing: Novel Inhibitors Attenuate Virulence in Staphylococcus aureus and Pseudomonas aeruginosa

靶向自诱导物-2群体感应:新型抑制剂减弱金黄色葡萄球菌和铜绿假单胞菌的毒力

Pellegrini, Angelica; Milli, Giorgio; Bellan Menegussi, Elisa; Viglio, Simona; Cinaglia, Pietro; Listro, Roberta; Linciano, Pasquale; Collina, Simona; Pietrocola, Giampiero

Screening macrocyclic peptide libraries by yeast display allows control of selection process and affinity ranking.

利用酵母展示技术筛选大环肽库可以控制选择过程和亲和力排序

Linciano Sara, Mazzocato Ylenia, Romanyuk Zhanna, Vascon Filippo, Farrera-Soler Lluc, Will Edward, Xing Yuyu, Chen Shiyu, Kumada Yoichi, Simeoni Marta, Scarso Alessandro, Cendron Laura, Heinis Christian, Angelini Alessandro

HuR-Targeted Small Molecules Reduce Pseudomonas aeruginosa Adhesion in Cystic Fibrosis Airway Epithelial Cells

靶向HuR的小分子可降低铜绿假单胞菌在囊性纤维化气道上皮细胞中的黏附

Listro, Roberta; Pellegrini, Angelica; Rossino, Giacomo; Linciano, Pasquale; Pietrocola, Giampiero; Collina, Simona

1,3-Dithiolane as a Privileged Scaffold in Bioactive Derivatives: Chiral Resolution and Assignment of Absolute Configuration

1,3-二硫杂环戊烷作为生物活性衍生物中的优势骨架:手性拆分和绝对构型确定

Listro, Roberta; Rossino, Giacomo; Cavalloro, Valeria; Rossi, Daniela; Boiocchi, Massimo; Robescu, Marina Simona; Bavaro, Teodora; Franchini, Silvia; Sorbi, Claudia; De Amici, Marco; Linciano, Pasquale; Collina, Simona

Neurodegeneration: can metabolites from Eremurus persicus help?

神经退行性疾病:Eremurus persicus 的代谢物有帮助吗?

Cavalloro, Valeria; Marchesi, Nicoletta; Linciano, Pasquale; Rossi, Daniela; Campagnoli, Lucrezia Irene Maria; Fossati, Alice; Ahmed, Karzan Mahmood; Malacrida, Alessio; Miloso, Mariarosaria; Mazzeo, Giuseppe; Abbate, Sergio; Longhi, Giovanna; Ambrosio, Francesca Alessandra; Costa, Giosuè; Alcaro, Stefano; Pascale, Alessia; Martino, Emanuela; Collina, Simona

Crystal structure of human serum albumin in complex with megabody reveals unique human and murine cross-reactive binding site

人血清白蛋白与巨抗体复合物的晶体结构揭示了独特的人类和鼠交叉反应结合位点

Sofia De Felice, Zhanna Romanyuk, Monica Chinellato, Giulia Zoia, Sara Linciano, Yoichi Kumada, Els Pardon, Jan Steyaert, Alessandro Angelini, Laura Cendron

Peptide Nucleic Acids in Saturation Transfer Difference Nuclear Magnetic Resonance Experiments: A Simple and Valuable Tool for Studying HuR-Small Molecule Complexes

肽核酸在饱和转移差分核磁共振实验中的应用:研究HuR-小分子复合物的简单而有价值的工具

Gado, Irene; Garbagnoli, Martina; Ambrosio, Francesca Alessandra; Listro, Roberta; Parafioriti, Michela; Cauteruccio, Silvia; Rossi, Daniela; Linciano, Pasquale; Costa, Giosuè; Alcaro, Stefano; Vasile, Francesca; Collina, Simona

Biophysical Assays for Investigating Modulators of Macromolecular Complexes: An Overview

用于研究大分子复合物调节剂的生物物理分析:概述

Garbagnoli, Martina; Linciano, Pasquale; Listro, Roberta; Rossino, Giacomo; Vasile, Francesca; Collina, Simona

A green Heck reaction protocol towards trisubstituted alkenes, versatile pharmaceutical intermediates

针对三取代烯烃、多功能药物中间体的绿色 Heck 反应方案

Giacomo Rossino, Giorgio Marrubini, Margherita Brindisi, Marc Granje, Pasquale Linciano, Daniela Rossi, Simona Collina