日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

A pan-respiratory antiviral chemotype targeting a transient host multi-protein complex

一种靶向瞬时宿主多蛋白复合物的泛呼吸道抗病毒化学型

Michon, Maya; Müller-Schiffmann, Andreas; Lingappa, Anuradha F; Yu, Shao Feng; Du, Li; Deiter, Fred; Broce, Sean; Mallesh, Suguna; Crabtree, Jackelyn; Lingappa, Usha F; Macieik, Amanda; Müller, Lisa; Ostermann, Philipp Niklas; Andrée, Marcel; Adams, Ortwin; Schaal, Heiner; Hogan, Robert J; Tripp, Ralph A; Appaiah, Umesh; Anand, Sanjeev K; Campi, Thomas W; Ford, Michael J; Reed, Jonathan C; Lin, Jim; Akintunde, Olayemi; Copeland, Kiel; Nichols, Christine; Petrouski, Emma; Moreira, Ana R; Jiang, I-Ting; DeYarman, Nicholas; Brown, Ian; Lau, Sharon; Segal, Ilana; Goldsmith, Danielle; Hong, Shi; Asundi, Vinod; Briggs, Erica M; Phyo, Ngwe Sin; Froehlich, Markus; Onisko, Bruce; Matlack, Kent; Dey, Debendranath; Lingappa, Jaisri R; Prasad, Dharma M; Kitaygorodskyy, Anatoliy; Solas, Dennis; Boushey, Homer; Greenland, John; Pillai, Satish; Lo, Michael K; Montgomery, Joel M; Spiropoulou, Christina F; Korth, Carsten; Selvarajah, Suganya; Paulvannan, Kumar; Lingappa, Vishwanath R

Small molecule protein assembly modulators with pan-cancer therapeutic efficacy

具有泛癌治疗功效的小分子蛋白质组装调节剂

Lingappa, Anuradha F; Akintunde, Olayemi; Samueli, Erin; Ewald, Connie; Michon, Maya; Ziari, Niloufar; Lu, Ming; Yu, Shao Feng; Froehlich, Markus; Le, Phuong Uyen; Fernandez, Yuniel; Mallesh, Suguna; Lin, Jim; Kitaygorodskyy, Anatoliy; Solas, Dennis; Reed, Jonathan C; Lingappa, Jaisri R; Müller-Schiffmann, Andreas; Korth, Carsten; Prasad, Dharma; Nalca, Aysegul; Aston, Emily; Fabbri, Brad; Anand, Sanjeev K; Campi, Thomas W; Petrouski, Emma; Dey, Debendranath; Andrews, David W; Rubenstein, James L; Lingappa, Vishwanath R

Protein Assembly Modulation: A New Approach to Amyotrophic Lateral Sclerosis (ALS) Therapeutics

蛋白质组装调控:肌萎缩侧索硬化症(ALS)治疗的新方法

Yu, Shao Feng; Paulvannan, Kumar; Solas, Dennis; Lingappa, Anuradha F; Moreira, Ana Raquel; Sahu, Shriya; Michon, Maya; Macieik, Amanda; Goldsmith, Danielle; DeYarman, Nicholas; Mallesh, Suguna; Prasad, M Dharma; Maios, Claudia; Ruan, Kai; Tomassy, Giulio S; Jensen, Elizabeth; McGuirk, Emma; Bader, Verian; Mueller-Schiffmann, Andreas; Reed, Jonathan C; Lingappa, Jaisri R; Asundi, Vinod; Hong, Shi; Jacobsen, Steve; Brandon, Nicholas; Ostrow, Lyle; Lloyd, Tom; Parker, J Alex; Staats, Kim A; Ichida, Justin; Dodge, James C; Dey, Debendranath; Korth, Carsten; Selvarajah, Suganya; Lingappa, Vishwanath R; Rosenfeld, Jeffrey

A Pan-Respiratory Antiviral Chemotype Targeting a Host Multi-Protein Complex

一种靶向宿主多蛋白复合物的泛呼吸道抗病毒化学类型

Michon, Maya; Müller-Schiffmann, Andreas; Lingappa, Anuradha F; Yu, Shao Feng; Du, Li; Deiter, Fred; Broce, Sean; Mallesh, Suguna; Crabtree, Jackelyn; Lingappa, Usha F; Macieik, Amanda; Müller, Lisa; Ostermann, Philipp Niklas; Andrée, Marcel; Adams, Ortwin; Schaal, Heiner; Hogan, Robert J; Tripp, Ralph A; Appaiah, Umesh; Anand, Sanjeev K; Campi, Thomas W; Ford, Michael J; Reed, Jonathan C; Lin, Jim; Akintunde, Olayemi; Copeland, Kiel; Nichols, Christine; Petrouski, Emma; Moreira, A Raquel; Jiang, I-Ting; DeYarman, Nicholas; Brown, Ian; Lau, Sharon; Segal, Ilana; Goldsmith, Danielle; Hong, Shi; Asundi, Vinod; Briggs, Erica M; Phyo, Ngwe Sin; Froehlich, Markus; Onisko, Bruce; Matlack, Kent; Dey, Debendranath; Lingappa, Jaisri R; Prasad, M Dharma; Kitaygorodskyy, Anatoliy; Solas, Dennis; Boushey, Homer; Greenland, John; Pillai, Satish; Lo, Michael K; Montgomery, Joel M; Spiropoulou, Christina F; Korth, Carsten; Selvarajah, Suganya; Paulvannan, Kumar; Lingappa, Vishwanath R

Identification of an Antiretroviral Small Molecule That Appears To Be a Host-Targeting Inhibitor of HIV-1 Assembly

鉴定出一种抗逆转录病毒小分子,该分子似乎是一种针对宿主的 HIV-1 组装抑制剂

Jonathan C Reed, Dennis Solas, Anatoliy Kitaygorodskyy, Beverly Freeman, Dylan T B Ressler, Daryl J Phuong, J Victor Swain, Kent Matlack, Clarence R Hurt, Vishwanath R Lingappa, Jaisri R Lingappa

Addressing Antiretroviral Drug Resistance with Host-Targeting Drugs-First Steps towards Developing a Host-Targeting HIV-1 Assembly Inhibitor

利用宿主靶向药物解决抗逆转录病毒药物耐药性问题——开发宿主靶向HIV-1组装抑制剂的第一步

Lingappa, Jaisri R; Lingappa, Vishwanath R; Reed, Jonathan C

Formation of RNA Granule-Derived Capsid Assembly Intermediates Appears To Be Conserved between Human Immunodeficiency Virus Type 1 and the Nonprimate Lentivirus Feline Immunodeficiency Virus

RNA颗粒衍生衣壳组装中间体的形成在人类免疫缺陷病毒1型和非灵长类慢病毒猫免疫缺陷病毒之间似乎是保守的

Jonathan C Reed ,Nick Westergreen ,Brook C Barajas ,Dylan T B Ressler ,Daryl J Phuong ,John V Swain ,Vishwanath R Lingappa ,Jaisri R Lingappa

Assembly of immature HIV-1 capsids using a cell-free system

利用无细胞系统组装未成熟的HIV-1衣壳

Lingappa, Jaisri R; Thielen, Beth K

T cells contain an RNase-insensitive inhibitor of APOBEC3G deaminase activity.

T 细胞含有对 RNase 不敏感的 APOBEC3G 脱氨酶活性抑制剂

Thielen Beth K, Klein Kevin C, Walker Lorne W, Rieck Mary, Buckner Jane H, Tomblingson Garrett W, Lingappa Jaisri R