日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Monoclonal antibody inhibition of PAR2 reduces phenotype severity and pain in murine inflammatory bowel disease

单克隆抗体抑制PAR2可减轻小鼠炎症性肠病的表型严重程度和疼痛。

Ritoux, Anne; Grundy, Laura J; Manjappa, Pravallika; Paine, Luke W; Neisen, Jessica; Linley, John E; Smith, Ewan St John

SLC45A4 is a pain gene encoding a neuronal polyamine transporter

SLC45A4 是一种疼痛基因,编码神经元多胺转运蛋白。

Middleton, Steven J; Markússon, Sigurbjörn; Åkerlund, Mikael; Deme, Justin C; Tseng, Mandy; Li, Wenqianglong; Zuberi, Sana R; Kuteyi, Gabriel; Sarkies, Peter; Baskozos, Georgios; Perez-Sanchez, Jimena; Farah, Adham; Hébert, Harry L; Toikumo, Sylvanus; Yu, Zhanru; Maxwell, Susan; Dong, Yin Y; Kessler, Benedikt M; Kranzler, Henry R; Linley, John E; Smith, Blair H; Lea, Susan M; Parker, Joanne L; Lyssenko, Valeriya; Newstead, Simon; Bennett, David L

Efficacy of MEDI0618, a pH-dependent monoclonal antibody targeting PAR2, in preclinical models of migraine.

MEDI0618 是一种 pH 依赖性单克隆抗体,靶向 PAR2,在偏头痛的临床前模型中疗效

Kopruszinski Caroline M, Linley John E, Thornton Peter, Walker Alison S, Newton Philip, Podichetty Sadhana, Ruparel Radhey Hemendra, Moreira de Souza Luiz Henrique, Navratilova Edita, Meno-Tetang Guy, Gurrell Ian, Dodick David W, Dobson Claire, Chessell Tharani, Porreca Frank, Chessell Iain

Pain in fibrous dysplasia: identifying nociceptive mechanisms in a preclinical model

纤维性骨发育不良中的疼痛:在临床前模型中识别伤害感受机制

Hopkins, Chelsea; de Castro, Luis Fernandez; Benthin, Julie; Diaz-delCastillo, Marta; Manjappa, Pravallika; Boyce, Alison; Mendoza, Ruth Elena Martinez; Mora, Juan Antonio Vazquez; Lopez-Delgado, Giovanni Emmanuel; Gomez, Lizeth Yazmin Ponce; Mohamed, Khaled Elhady; Linley, John E; Collins, Michael T; Jimenez-Andrade, Juan Miguel; Heegaard, Anne-Marie

Identification of SLC45A4 as a pain gene encoding a neuronal polyamine transporter

鉴定出 SLC45A4 为编码神经元多胺转运蛋白的疼痛基因

Middleton, Steven J; Markússon, Sigurbjörn; Åkerlund, Mikael; Deme, Justin C; Tseng, Mandy; Li, Wenqianglong; Zuberi, Sana R; Kuteyi, Gabriel; Sarkies, Peter; Baskozos, Georgios; Perez-Sanchez, Jimena; Hébert, Harry L; Toikumo, Sylvanus; Farah, Adham; Maxwell, Susan; Dong, Yin Y; Kranzler, Henry R; Linley, John E; Smith, Blair H; Lea, Susan M; Parker, Joanne L; Lyssenko, Valeriya; Newstead, Simon; Bennett, David L

Pregabalin Silences Oxaliplatin-Activated Sensory Neurons to Relieve Cold Allodynia.

普瑞巴林抑制奥沙利铂激活的感觉神经元,从而缓解寒冷性痛觉过敏

Iseppon Federico, Luiz Ana P, Linley John E, Wood John N

Calcium imaging for analgesic drug discovery

钙成像技术在镇痛药物研发中的应用

Iseppon, Federico; Linley, John E; Wood, John N

Bradykinin controls pool size of sensory neurons expressing functional δ-opioid receptors

缓激肽控制表达功能性δ-阿片受体的感觉神经元的数量。

Pettinger, Louisa; Gigout, Sylvain; Linley, John E; Gamper, Nikita

Neurological perspectives on voltage-gated sodium channels

电压门控钠通道的神经学视角

Eijkelkamp, Niels; Linley, John E; Baker, Mark D; Minett, Michael S; Cregg, Roman; Werdehausen, Robert; Rugiero, François; Wood, John N

TRPC3 and TRPC6 are essential for normal mechanotransduction in subsets of sensory neurons and cochlear hair cells

TRPC3 和 TRPC6 对于部分感觉神经元和耳蜗毛细胞的正常机械转导至关重要。

Quick, Kathryn; Zhao, Jing; Eijkelkamp, Niels; Linley, John E; Rugiero, Francois; Cox, James J; Raouf, Ramin; Gringhuis, Martine; Sexton, Jane E; Abramowitz, Joel; Taylor, Ruth; Forge, Andy; Ashmore, Jonathan; Kirkwood, Nerissa; Kros, Corné J; Richardson, Guy P; Freichel, Marc; Flockerzi, Veit; Birnbaumer, Lutz; Wood, John N