日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Selective small molecule targeting of KDM4 as a therapeutic strategy to reduce proliferation of acute myeloid leukaemia

选择性小分子靶向KDM4作为减少急性髓系白血病增殖的治疗策略

Monaghan, Laura; Bunschoten, Roderick P; Bittencourt-Silvestre, Joana; Park, Taeju; Gannon, Susan; Pirvan, Petrisor Alin; Hoose, Alex; Wheadon, Helen; Liskamp, Robert M J; Huang, Xu; Jørgensen, Heather G

Orthogonal Covalent Entrapment of Cargo into Biodegradable Polymeric Micelles via Native Chemical Ligation

通过天然化学连接将货物正交共价包埋到可生物降解的聚合物胶束中

Hebels, Erik R; Bindt, Felix; Walther, Johanna; van Geijn, Michiel; Weterings, Jimmy; Hu, Qizhi; Colombo, Claudio; Liskamp, Rob; Rijcken, Cristianne; Hennink, Wim E; Vermonden, Tina

Versatile Click Linker Enabling Native Peptide Release from Nanocarriers upon Redox Trigger

多功能点击连接子可在氧化还原触发下从纳米载体中释放天然肽

Erik R Hebels ,Stefanie Dietl ,Matt Timmers ,Jaimie Hak ,Antionette van den Dikkenberg ,Cristianne J F Rijcken ,Wim E Hennink ,Rob M J Liskamp ,Tina Vermonden

Exploring the Chemical Properties and Medicinal Applications of Tetramethylthiocycloheptyne Sulfoximine Used in Strain-Promoted Azide-Alkyne Cycloaddition Reactions

探索四甲硫基环庚炔亚砜亚胺在应变促进叠氮化物-炔烃环加成反应中的化学性质和药用应用

Matt Timmers, Andi Kipper, Raphael Frey, Stef Notermans, Maksym Voievudskyi, Claire Wilson, Nina Hentzen, Michael Ringle, Clara Bovino, Bernhard Stump, Cristianne J F Rijcken, Tina Vermonden, Ingrid Dijkgraaf, Rob Liskamp

A New Class of Tunable Acid-Sensitive Linkers for Native Drug Release Based on the Trityl Protecting Group

基于三苯甲基保护基的新型可调酸敏连接子用于天然药物释放

Timmers, Matt; Weterings, Jimmy; van Geijn, Michiel; Bell, Roel; Lenting, Peter E; Rijcken, Cristianne J F; Vermonden, Tina; Hennink, Wim E; Liskamp, Rob M J

Excessive esophageal toxicity in patients with locally advanced non-small cell lung cancer treated with concurrent hypofractionated chemoradiotherapy and 3-weekly platinum doublet chemotherapy

局部晚期非小细胞肺癌患者接受同步低分割放化疗和每3周一次的铂类双药化疗后,出现过量食管毒性。

van der Voort van Zyp, Noëlle; Hashimzadah, Masoma; Kouwenhoven, Erik; Liskamp, Carmen; Gadellaa-van Hooijdonk, Christa; Pouw, Ellen; Belderbos, Jose; Maas, Klaartje; van de Vaart, Paul; Mast, Mirjam

A KDM4A-PAF1-mediated epigenomic network is essential for acute myeloid leukemia cell self-renewal and survival

KDM4A-PAF1 介导的表观基因组网络对于急性髓系白血病细胞的自我更新和存活至关重要

Matthew E Massett, Laura Monaghan, Shaun Patterson, Niamh Mannion, Roderick P Bunschoten, Alex Hoose, Sandra Marmiroli, Robert M J Liskamp, Heather G Jørgensen, David Vetrie, Alison M Michie, Xu Huang

Design and Synthesis of HCV-E2 Glycoprotein Epitope Mimics in Molecular Construction of Potential Synthetic Vaccines

HCV-E2 糖蛋白表位模拟物的设计和合成及其在潜在合成疫苗分子构建中的应用

Theodorus J Meuleman, Vanessa M Cowton, Arvind H Patel, Rob M J Liskamp

TMTHSI, a superior 7-membered ring alkyne containing reagent for strain-promoted azide-alkyne cycloaddition reactions

TMTHSI 是一种优良的含七元环炔烃的试剂,适用于应变促进的叠氮-炔环加成反应。

Weterings, Jimmy; Rijcken, Cristianne J F; Veldhuis, Harald; Meulemans, Tommi; Hadavi, Darya; Timmers, Matt; Honing, Maarten; Ippel, Hans; Liskamp, Rob M J

Nodal recurrence patterns on PET/CT after RTOG-based nodal radiotherapy for prostate cancer

前列腺癌RTOG方案淋巴结放疗后PET/CT显示的淋巴结复发模式

Liskamp, C P; Donswijk, M L; van der Poel, H G; Schaake, E E; Vogel, W V