日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

BRAF(V600E)-Driven Lung Tumorigenesis Requires Ligand-Mediated Activation of ERBB Receptor Signaling.

BRAF(V600E)驱动的肺肿瘤发生需要配体介导的ERBB受体信号激活

Dacheux Melanie Angelina, Wu Meng-Jung, Scherzer Michael T, Nillson Monique, Murphy Brandon, Schuman Sophia, Ju Zhenlin, Bivona Trever, Lito Piro, Gumbleton Matthew, Puri Sonam, Akerley Wallace, Wang Jing, Wang Kaiwen, Heymach John, Kinsey Conan G, Negrao Marcelo, McMahon Martin, Vaishnavi Aria

Preclinical Evaluation of [(124)I]-Sotorasib for the Imaging of Kirsten Rat Sarcoma G12C Mutant Tumors.

[(124)I]-Sotorasib 用于 Kirsten 大鼠肉瘤 G12C 突变肿瘤成像的临床前评价

Artschwager Raik, Kalidindi Teja M, Johnson Delissa, Brennan Christopher, Samuels Zachary V, Lito Piro, Pillarsetty Naga Vara Kishore

Chemical remodeling of a cellular chaperone to target the active state of mutant KRAS

通过化学方法改造细胞伴侣蛋白,使其靶向突变型KRAS的活性状态

Schulze, Christopher J; Seamon, Kyle J; Zhao, Yulei; Yang, Yu C; Cregg, Jim; Kim, Dongsung; Tomlinson, Aidan; Choy, Tiffany J; Wang, Zhican; Sang, Ben; Pourfarjam, Yasin; Lucas, Jessica; Cuevas-Navarro, Antonio; Ayala-Santos, Carlos; Vides, Alberto; Li, Chuanchuan; Marquez, Abby; Zhong, Mengqi; Vemulapalli, Vidyasiri; Weller, Caroline; Gould, Andrea; Whalen, Daniel M; Salvador, Anthony; Milin, Anthony; Saldajeno-Concar, Mae; Dinglasan, Nuntana; Chen, Anqi; Evans, Jim; Knox, John E; Koltun, Elena S; Singh, Mallika; Nichols, Robert; Wildes, David; Gill, Adrian L; Smith, Jacqueline A M; Lito, Piro

Long-Term Outcomes and Molecular Correlates of Sotorasib Efficacy in Patients With Pretreated KRAS G12C-Mutated Non-Small-Cell Lung Cancer: 2-Year Analysis of CodeBreaK 100

索托拉西布治疗既往接受过治疗的KRAS G12C突变型非小细胞肺癌患者的长期疗效及分子相关性:CodeBreak 100研究的2年分析

Dy, Grace K; Govindan, Ramaswamy; Velcheti, Vamsidhar; Falchook, Gerald S; Italiano, Antoine; Wolf, Jürgen; Sacher, Adrian G; Takahashi, Toshiaki; Ramalingam, Suresh S; Dooms, Christophe; Kim, Dong-Wan; Addeo, Alfredo; Desai, Jayesh; Schuler, Martin; Tomasini, Pascale; Hong, David S; Lito, Piro; Tran, Qui; Jones, Simon; Anderson, Abraham; Hindoyan, Antreas; Snyder, Wendy; Skoulidis, Ferdinandos; Li, Bob T

Clinical and Genomic Features of Response and Toxicity to Sotorasib in a Real-World Cohort of Patients With Advanced KRAS G12C-Mutant Non-Small Cell Lung Cancer

在真实世界队列中,Sotorasib治疗晚期KRAS G12C突变型非小细胞肺癌患者的临床和基因组学特征及其疗效和毒性

Thummalapalli, Rohit; Bernstein, Ezra; Herzberg, Benjamin; Li, Bob T; Iqbal, Afsheen; Preeshagul, Isabel; Santini, Fernando C; Eng, Juliana; Ladanyi, Marc; Yang, Soo-Ryum; Shen, Ronglai; Lito, Piro; Riely, Gregory J; Sabari, Joshua K; Arbour, Kathryn C

Outcomes of Combination Platinum-Doublet Chemotherapy and Anti-PD(L)-1 Blockade in KRASG12C-Mutant Non-Small Cell Lung Cancer

铂类双药化疗联合抗PD(L)-1阻断治疗KRASG12C突变型非小细胞肺癌的疗效

Elkrief, Arielle; Riccuiti, Biagio; Alessi, Joao V; Fei, Teng; Kalvin, Hannah L; Egger, Jacklynn V; Rizvi, Hira; Thummalapalli, Rohit; Lamberti, Guiseppe; Plodkowski, Andrew; Hellmann, Matthew D; Kris, Mark G; Arcila, Maria E; Baine, Marina K; Rudin, Charles M; Lito, Piro; Ladanyi, Marc; Schoenfeld, Adam J; Riely, Gregory J; Awad, Mark M; Arbour, Kathryn C

Overall survival with circulating tumor DNA-guided therapy in advanced non-small-cell lung cancer

循环肿瘤DNA指导治疗晚期非小细胞肺癌的总体生存率

Jee, Justin; Lebow, Emily S; Yeh, Randy; Das, Jeeban P; Namakydoust, Azadeh; Paik, Paul K; Chaft, Jamie E; Jayakumaran, Gowtham; Rose Brannon, A; Benayed, Ryma; Zehir, Ahmet; Donoghue, Mark; Schultz, Nikolaus; Chakravarty, Debyani; Kundra, Ritika; Madupuri, Ramyasree; Murciano-Goroff, Yonina R; Tu, Hai-Yan; Xu, Chong-Rui; Martinez, Andrés; Wilhelm, Clare; Galle, Jesse; Daly, Bobby; Yu, Helena A; Offin, Michael; Hellmann, Matthew D; Lito, Piro; Arbour, Kathryn C; Zauderer, Marjorie G; Kris, Mark G; Ng, Kenneth K; Eng, Juliana; Preeshagul, Isabel; Victoria Lai, W; Fiore, John J; Iqbal, Afsheen; Molena, Daniela; Rocco, Gaetano; Park, Bernard J; Lim, Lee P; Li, Mark; Tong-Li, Candace; De Silva, Madhawa; Chan, David L; Diakos, Connie I; Itchins, Malinda; Clarke, Stephen; Pavlakis, Nick; Lee, Adrian; Rekhtman, Natasha; Chang, Jason; Travis, William D; Riely, Gregory J; Solit, David B; Gonen, Mithat; Rusch, Valerie W; Rimner, Andreas; Gomez, Daniel; Drilon, Alexander; Scher, Howard I; Shah, Sohrab P; Berger, Michael F; Arcila, Maria E; Ladanyi, Marc; Levine, Ross L; Shen, Ronglai; Razavi, Pedram; Reis-Filho, Jorge S; Jones, David R; Rudin, Charles M; Isbell, James M; Li, Bob T

Immune biomarkers and response to checkpoint inhibition of BRAF(V600) and BRAF non-V600 altered lung cancers

BRAF(V600)和BRAF非V600突变肺癌的免疫生物标志物及对检查点抑制剂的反应

Murciano-Goroff, Yonina R; Pak, Terry; Mondaca, Sebastian; Flynn, Jessica R; Montecalvo, Joseph; Rekhtman, Natasha; Halpenny, Darragh; Plodkowski, Andrew J; Wu, Stephanie L; Kris, Mark G; Paik, Paul K; Riely, Gregory J; Yu, Helena A; Rudin, Charles M; Hellmann, Matthew D; Land, Josiah D; Buie, Larry W; Heller, Glenn; Lito, Piro; Yaeger, Rona; Drilon, Alexander; Liu, Dazhi; Li, Bob T; Offin, Michael

Phase 1 Clinical Trial of Trametinib and Ponatinib in Patients With NSCLC Harboring KRAS Mutations

Trametinib 和 Ponatinib 治疗携带 KRAS 突变的非小细胞肺癌患者的 I 期临床试验

Arbour, Kathryn C; Manchado, Eusebio; Bott, Matthew J; Ahn, Linda; Tobi, Yosef; Ni, Andy Ai; Yu, Helena A; Shannon, Alyssa; Ladanyi, Marc; Perron, Victoria; Ginsberg, Michelle S; Johnson, Amanda; Holodny, Andrei; Kris, Mark G; Rudin, Charles M; Lito, Piro; Rosen, Neal; Lowe, Scott; Riely, Gregory J

Acquired Resistance to KRAS(G12C) Inhibition in Cancer

癌症中对KRAS(G12C)抑制剂的获得性耐药

Awad, Mark M; Liu, Shengwu; Rybkin, Igor I; Arbour, Kathryn C; Dilly, Julien; Zhu, Viola W; Johnson, Melissa L; Heist, Rebecca S; Patil, Tejas; Riely, Gregory J; Jacobson, Joseph O; Yang, Xiaoping; Persky, Nicole S; Root, David E; Lowder, Kristen E; Feng, Hanrong; Zhang, Shannon S; Haigis, Kevin M; Hung, Yin P; Sholl, Lynette M; Wolpin, Brian M; Wiese, Julie; Christiansen, Jason; Lee, Jessica; Schrock, Alexa B; Lim, Lee P; Garg, Kavita; Li, Mark; Engstrom, Lars D; Waters, Laura; Lawson, J David; Olson, Peter; Lito, Piro; Ou, Sai-Hong I; Christensen, James G; Jänne, Pasi A; Aguirre, Andrew J