日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Enhancing schistosomiasis drug discovery approaches with optimized proteasome substrates.

利用优化的蛋白酶体底物增强血吸虫病药物发现方法

Silva Elany B, Jiang Zhenze, Liu Chenxi, Fajtová Pavla, Teixeira Thaiz R, de Castro Fiorini Maia Giovana, Liu Lawrence J, El-Sakkary Nelly, Skinner Danielle E, Syed Ali, Wang Steven C, Caffrey Conor R, O'Donoghue Anthony J

An in vitro platform for the enzymatic characterization of the rhomboid protease RHBDL4

用于菱形蛋白酶RHBDL4酶学表征的体外平台

Bhaduri, Satarupa; Braza, Mac Kevin E; Stanchev, Stancho; Tauber, Marina; Al-Bawab, Raghad; Liu, Lawrence J; Trujillo, Diego F; Solorio-Kirpichyan, Kristina; Srivastava, Ambuj; Sanlley-Hernandez, Javier; O'Donoghue, Anthony J; Lemberg, Marius K; Amaro, Rommie; Strisovsky, Kvido; Neal, Sonya E

Discovery of small molecules with anthelmintic potential in the Medicines for Malaria Venture's COVID and Global Health Priority Boxes using an infrared-based assay for Caenorhabditis elegans motility

利用基于红外光谱的秀丽隐杆线虫运动性检测方法,在疟疾药物研发联盟的COVID-19和全球健康优先项目箱中发现具有抗蠕虫潜力的分子。

Sun, Yujie Uli; Liu, Lawrence J; Caffrey, Conor R

Distinct substrate specificities of the three catalytic subunits of the Trichomonas vaginalis proteasome.

阴道毛滴虫蛋白酶体的三个催化亚基具有不同的底物特异性

Fajtova Pavla, Hurysz Brianna M, Miyamoto Yukiko, Serafim Mateus Sá M, Jiang Zhenze, Vazquez Julia M, Trujillo Diego F, Liu Lawrence J, Somani Urvashi, Almaliti Jehad, Myers Samuel A, Caffrey Conor R, Gerwick William H, McMinn Dustin L, Kirk Christopher J, Boura Evzen, Eckmann Lars, O'Donoghue Anthony J

Structure activity relationships of antischistosomal N-phenylbenzamides by incorporation of electron-withdrawing functionalities

通过引入吸电子基团研究抗血吸虫N-苯基苯甲酰胺的构效关系

Dawoodjee, Ameera Mohammed; Sichinga, John; Banda, Harrison; Mbaya, Steve; Funjika, Evelyn; Mayoka, Godfrey; Hikaambo, Christabel; Francisco, Karol R; Sun, Yujie Uli; Liu, Lawrence J; Caffrey, Conor R; Cheuka, Peter Mubanga

Design, Synthesis, and Evaluation of An Anti-trypanosomal [1,2,4]Triazolo[1,5-a]pyrimidine Probe for Photoaffinity Labeling Studies.

设计、合成和评价抗锥虫[1,2,4]三唑并[1,5-a]嘧啶探针用于光亲和标记研究

Lucero Bobby, Francisco Karol R, Varricchio Carmine, Liu Lawrence J, Yao Yuemang, Brancale Andrea, Brunden Kurt R, Caffrey Conor R, Ballatore Carlo

An in vitro platform for the enzymatic characterization of the rhomboid protease RHBDL4

用于菱形蛋白酶RHBDL4酶学表征的体外平台

Bhaduri, Satarupa; Braza, Mac Kevin E; Stanchev, Stancho; Tauber, Marina; Al-Bawab, Raghad; Liu, Lawrence J; Trujillo, Diego F; Solorio-Kirpichyan, Kristina; Srivastava, Ambuj; Sanlley-Hernandez, Javier; O'Donoghue, Anthony J; Lemberg, Marius K; Amario, Rommie; Strisovsky, Kvido; Neal, Sonya E

Structure-activity relationship of dibenzylideneacetone analogs against the neglected disease pathogen, Trypanosoma brucei

二亚苄基丙酮类似物对被忽视的病原体布氏锥虫的构效关系

Francisco, Karol R; Monti, Ludovica; Yang, Wenqian; Park, Hayoung; Liu, Lawrence J; Watkins, Kaitlyn; Amarasinghe, Dilini K; Nalli, Marianna; Roberto Polaquini, Carlos; Regasini, Luis O; Eduardo Miller Crotti, Antônio; Silvestri, Romano; Guidi Magalhães, Lizandra; Caffrey, Conor R

Activity of N-phenylbenzamide analogs against the neglected disease pathogen, Schistosoma mansoni

N-苯基苯甲酰胺类似物对被忽视的病原体曼氏血吸虫的活性

Kanyanta, Masebe; Lengwe, Chilufya; Mambwe, Dickson; Francisco, Karol R; Liu, Lawrence J; Uli Sun, Yujie; Amarasinghe, Dilini K; Caffrey, Conor R; Mubanga Cheuka, Peter

Identification of a role for CLASP2 in insulin action

确定 CLASP2 在胰岛素作用中的作用

Paul Langlais, James L Dillon, April Mengos, Debra P Baluch, Ranna Ardebili, Danielle N Miranda, Xitao Xie, Bradlee L Heckmann, Jun Liu, Lawrence J Mandarino