日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

High-Throughput Screening of Potent Drug-like Molecules Targeting 17β-HSD10 for the Treatment of Alzheimer's Disease and Cancer

利用高通量筛选靶向17β-HSD10的强效类药分子,用于治疗阿尔茨海默病和癌症

Aitken, Laura; Baillie, Gemma; Pannifer, Andrew; Morrison, Angus; Major, Louise L; Alphey, Magnus S; Sethi, Ritika; Timmerman, Martin; Robinson, John; Riley, Jennifer; Shishikura, Yoko; Koekemoer, Lizbe; Von Delft, Frank; Rutjes, Helma; Read, Kevin D; Jones, Philip S; McElroy, Stuart P; Smith, Terry K; Gunn-Moore, Frank J

Crystallographic Fragment Screen of Coxsackievirus A16 2A Protease identifies new opportunities for the development of broad-spectrum anti-enterovirals

柯萨奇病毒A16 2A蛋白酶的晶体学片段筛选为开发广谱抗肠道病毒药物提供了新的契机

Lithgo, Ryan M; Tomlinson, Charles W E; Fairhead, Michael; Winokan, Max; Thompson, Warren; Wild, Conor; Aschenbrenner, Jasmin Cara; Balcomb, Blake H; Marples, Peter G; Chandran, Anu V; Golding, Mathew; Koekemoer, Lizbe; Williams, Eleanor P; Wang, SiYl; Ni, Xiaomin; MacLean, Elizabeth; Giroud, Charline; Godoy, Andre Schutzer; Xavier, Mary-Ann; Walsh, Martin; Fearon, Daren; von Delft, Frank

Identifying novel chemical matter against the Chikungunya virus nsP3 macrodomain through crystallographic fragment screening

通过晶体学片段筛选鉴定针对基孔肯雅病毒nsP3宏结构域的新型化学物质

Aschenbrenner, Jasmin C; de Godoy, Andre Schutzer; Fairhead, Michael; Tomlinson, Charles W E; Winokan, Max; Balcomb, Blake H; Capkin, Eda; Chandran, Anu V; Golding, Mathew; Koekemoer, Lizbe; Lithgo, Ryan M; Marples, Peter G; Ni, Xiaomin; Thompson, Warren; Wild, Conor; Xavier, Mary-Ann E; Fearon, Daren; von Delft, Frank