Identification and evaluation of small-molecule inhibitors against the dNTPase SAMHD1 via a comprehensive screening funnel
通过综合筛选流程鉴定和评价针对 dNTPase SAMHD1 的小分子抑制剂
期刊:iScience
影响因子:4.6
doi:10.1016/j.isci.2024.108907
Si Min Zhang ,Cynthia B J Paulin ,Huazhang Shu ,Miriam Yagüe-Capilla ,Maurice Michel ,Petra Marttila ,Florian Ortis ,Henri Colyn Bwanika ,Christopher Dirks ,Rajagopal Papagudi Venkatram ,Elisée Wiita ,Ann-Sofie Jemth ,Ingrid Almlöf ,Olga Loseva ,Femke M Hormann ,Tobias Koolmeister ,Erika Linde ,Sun Lee ,Sabin Llona-Minguez ,Martin Haraldsson ,Hanna Axelsson ,Kia Strömberg ,Evert J Homan ,Martin Scobie ,Thomas Lundbäck ,Thomas Helleday ,Sean G Rudd