日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

One-Pot Base-Free Suzuki-Miyaura [(11)C]Methylation: Kinetic and Mechanistic Insights

一锅法无碱Suzuki-Miyaura [(11)C]甲基化反应:动力学和机理研究

Moreno, Oscar; Azzeggarh, Imad; Holland, Jason P; Windhorst, Albert D; Llop, Jordi

A brain-penetrant P2X7R antagonist mitigates Alzheimer's disease pathology

一种能穿透血脑屏障的P2X7R拮抗剂可减轻阿尔茨海默病病理。

Turcu, Andreea L; Oken, Adam C; Griñán-Ferré, Christian; Durner, Anna; Sierra-Marquez, Juan; Hinz-Kowalik, Sonja; Nagel, Jessica; Lee, So-Deok; Tzortzini, Efpraxia; Georgiou, Kyriakos; Bhol, Mamina; Baz, Zuriñe; Llop, Jordi; Schneider, Marion; Barbaraci, Carla; Kim, Ga-Ram; Barniol-Xicota, Marta; Val, Cristina; Brea, José; Loza, M Isabel; Pérez, Belén; Naesens, Lieve; Kolocouris, Antonios; Kim, Yong-Chul; Müller, Christa E; Nicke, Annette; Pallàs, Mercè; Mansoor, Steven E; Vázquez, Santiago

Increased levels of GFAP and purinergic P2X7 receptor in Alzheimer's disease brain are associated with Aβ, tau pathologies and synaptic loss

阿尔茨海默病患者脑组织中GFAP和嘌呤能P2X7受体水平升高与Aβ、tau蛋白病变和突触丢失有关。

Maschio, Cinzia A; Moreno, Oscar; Wang, Junlong; Maheshwari, Upasana; Keller, Annika; Konietzko, Uwe; Razansky, Daniel; Nordberg, Agneta; Rominger, Axel; Hock, Christoph; Llop, Jordi; Nitsch, Roger M; Ni, Ruiqing

Synthetic heparan sulfate mimics based on chitosan derivatives show broad-spectrum antiviral activity.

基于壳聚糖衍生物的合成硫酸乙酰肝素类似物表现出广谱抗病毒活性

Revuelta Julia, Rusu Luciana, Frances-Gomez Clara, Trapero Elena, Iglesias Susana, Pinilla Eva Calvo, Blázquez Ana-Belén, Gutiérrez-Adán Alfonso, Konuparamban Acsah, Moreno Oscar, Gómez Martínez María, Forcada-Nadal Alicia, López-Redondo María Luisa, Avilés-Alía Ana Isabel, Llácer José Luis, Llop Jordi, Martín Acebes Miguel Ángel, Geller Ron, Fernández-Mayoralas Alfonso

Longitudinal imaging evaluation of the inflammatory role of purinergic A(2)A receptors during subacute and chronic ischemic stroke.

亚急性及慢性缺血性卒中期间嘌呤能 A(2)A 受体炎症作用的纵向影像学评估

Garbizu Maider, Mocha-Muñoz Naroa, Rubio-López Esther, Palacios Laura, Aguado Laura, Ardaya María, Joya Ana, Alduntzin Unai, Plaza-García Sandra, Padro Daniel, Gómez-Vallejo Vanessa, Cossío Unai, Higuchi Makoto, Ramos-Cabrer Pedro, Zugaza José Luis, Llop Jordi, Martín Abraham

Chronic treatment with adenosine A1 receptor antagonist promotes neurogenesis and improves outcome after cerebral ischemia.

长期使用腺苷 A1 受体拮抗剂可促进神经发生,改善脑缺血后的预后

Ardaya Maria, Benito-Muñoz Monica, Rubio-López Esther, Garbizu Maider, Aguado Laura, Mocha-Muñoz Naroa, Iglesias Leyre, Aldutzin Unai, Matute Carlos, Soria Federico N, Gómez-Vallejo Vanessa, García-Etxarri Aitzol, Llop Jordi, Cavaliere Fabio, Martín Abraham

Synthesis and PET Imaging Biodistribution Studies of Radiolabeled Iododiflunisal, a Transthyretin Tetramer Stabilizer, Candidate Drug for Alzheimer's Disease

放射性标记的碘二氟尼柳(一种转甲状腺素四聚体稳定剂,阿尔茨海默病候选药物)的合成及PET成像生物分布研究

Joshi, Sameer M; Wilson, Thomas C; Li, Zibo; Preshlock, Sean; Gómez-Vallejo, Vanessa; Gouverneur, Véronique; Llop, Jordi; Arsequell, Gemma

Lipidomics and biodistribution of extracellular vesicles-secreted by hepatocytes from Zucker lean and fatty rats

Zucker瘦鼠和肥胖鼠肝细胞分泌的细胞外囊泡的脂质组学和生物分布

Azparren-Angulo, Maria; Mleczko, Justyna; Alboniga, Oihane E; Kruglik, Sergei; Guigner, Jean-Michel; Gonzalez, Esperanza; Garcia-Vallicrosa, Clara; Llop, Jordi; Simó, Cristina; Alonso, Cristina; Iruarrizaga, Marta; Royo, Felix; Falcon-Perez, Juan M

Increased uptake of the P2X7 receptor radiotracer (18) F-JNJ-64413739 in the brain and peripheral organs according to the severity of status epilepticus in male mice

雄性小鼠癫痫持续状态严重程度与脑和外周器官中 P2X7 受体放射性示踪剂 (18) F-JNJ-64413739 的摄取量增加相关。

Morgan, James; Moreno, Oscar; Alves, Mariana; Baz, Zuriñe; Menéndez Méndez, Aida; Leister, Hanna; Melia, Ciara; Smith, Jonathon; Visekruna, Alexander; Nicke, Annette; Bhattacharya, Anindya; Ceusters, Marc; Henshall, David C; Gómez-Vallejo, Vanessa; Llop, Jordi; Engel, Tobias

Anti-seizure effects of JNJ-54175446 in the intra-amygdala kainic acid model of drug-resistant temporal lobe epilepsy in mice

JNJ-54175446 在小鼠杏仁核内注射红藻氨酸诱导的耐药性颞叶癫痫模型中的抗癫痫作用

Mamad, Omar; Heiland, Mona; Lindner, Andreas U; Hill, Thomas D M; Ronroy, Ronan M; Rentrup, Kilian; Sanz-Rodriguez, Amaya; Langa, Elena; Heller, Janosch P; Moreno, Oscar; Llop, Jordi; Bhattacharya, Anindya; Palmer, James A; Ceusters, Marc; Engel, Tobias; Henshall, David C