Small-molecule multi-targeted kinase inhibitor RGB-286638 triggers P53-dependent and -independent anti-multiple myeloma activity through inhibition of transcriptional CDKs
小分子多靶点激酶抑制剂 RGB-286638 通过抑制转录 CDK 触发 P53 依赖性和 P53 非依赖性抗多发性骨髓瘤活性
期刊:Leukemia
影响因子:12.8
doi:10.1038/leu.2013.194
D Cirstea, T Hideshima, L Santo, H Eda, Y Mishima, N Nemani, Y Hu, N Mimura, F Cottini, G Gorgun, H Ohguchi, R Suzuki, H Loferer, N C Munshi, K C Anderson, N Raje