Drug-Like Properties in Macrocycles above MW 1000: Backbone Rigidity versus Side-Chain Lipophilicity
分子量大于1000的大环化合物的类药性质:主链刚性与侧链亲脂性
期刊:Angewandte Chemie-International Edition
影响因子:16.9
doi:10.1002/anie.202004550
Furukawa, Akihiro; Schwochert, Joshua; Pye, Cameron R; Asano, Daigo; Edmondson, Quinn D; Turmon, Alexandra C; Klein, Victoria G; Ono, Satoshi; Okada, Okimasa; Lokey, R Scott