Modifications to 1-(4-(2-Bis(4-fluorophenyl)methyl)sulfinyl)alkyl Alicyclic Amines That Improve Metabolic Stability and Retain an Atypical DAT Inhibitor Profile
对 1-(4-(2-双(4-氟苯基)甲基)亚磺酰基)烷基脂环胺进行修饰,以提高其代谢稳定性并保持非典型 DAT 抑制剂特性
期刊:Journal of Medicinal Chemistry
影响因子:6.8
doi:10.1021/acs.jmedchem.3c02037
Okorom, Amarachi V; Camacho-Hernandez, Gisela Andrea; Salomon, Kristine; Lee, Kuo Hao; Ku, Therese C; Cao, Jianjing; Won, Sung Joon; Friedman, Jacob; Lam, Jenny; Paule, James; Rais, Rana; Klein, Benjamin; Xi, Zheng-Xiong; Shi, Lei; Loland, Claus J; Newman, Amy Hauck