Synthesis, pharmacology and preclinical evaluation of (11)C-labeled 1,3-dihydro-2H-benzo[d]imidazole-2-ones for imaging γ8-dependent transmembrane AMPA receptor regulatory protein
利用 (11)C 标记的 1,3-二氢-2H-苯并[d]咪唑-2-酮进行 γ8 依赖性跨膜 AMPA 受体调节蛋白成像的合成、药理学和临床前评价
期刊:European Journal of Medicinal Chemistry
影响因子:5.9
doi:10.1016/j.ejmech.2018.08.019
Chen, Zhen; Mori, Wakana; Zhang, Xiaofei; Yamasaki, Tomoteru; Dunn, Patrick J; Zhang, Genwei; Fu, Hualong; Shao, Tuo; Zhang, Yiding; Hatori, Akiko; Ma, Longle; Fujinaga, Masayuki; Xie, Lin; Deng, Xiaoyun; Li, Hua; Yu, Qingzhen; Rong, Jian; Josephson, Lee; Ma, Jun-An; Shao, Yihan; Tomita, Susumu; Zhang, Ming-Rong; Liang, Steven H