日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Discovery of Small-Molecule Ligands for the E3 Ligase STUB1/CHIP from a DNA-Encoded Library Screen

从DNA编码文库筛选中发现E3连接酶STUB1/CHIP的小分子配体

Lucas, Simon C C; Milbradt, Alexander G; Breed, Jason; De Genst, Erwin; Jackson, Anne; Solovyeva, Alisa; Ackroyd, Bryony; Bauer, Matthias R; Liu, Juntai; Longmire, David; Petrović, Dušan; Rivers, Emma L; Stubbs, Christopher; Winlow, Poppy; Bazzaz, Sana; Dickson, Paige; Gikunju, Diana; Guié, Marie-Aude; Guilinger, John P; Hupp, Christopher D; Jetson, Rachael; Keefe, Anthony D; Nugai, Katherine; Yeoman, John T S; Zhang, Ying; Feng, Xian; Yu, Dequan; Phillips, Christopher

A high-throughput compatible workflow for the biochemical identification and characterization of molecular glues.

用于分子胶的生化鉴定和表征的高通量兼容工作流程

Guilbert Ryan, Couturier Maxime, Si Yuanyuan, Donovan Daniel O', Longmire David, Mak Hazel, Clarkson Paul, Argyrou Argyrides

Lipidated Stapled Peptides Targeting the Acyl Binding Protein UNC119

靶向酰基结合蛋白UNC119的脂化交联肽

Cromm, Philipp M; Adihou, Hélène; Kapoor, Shobhna; Vazquez-Chantada, Mercedes; Davey, Paul; Longmire, David; Hennes, Elisabeth; Hofer, Walter; Küchler, Philipp; Chiarparin, Elisabetta; Waldmann, Herbert; Grossmann, Tom N