日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Novel binding mode for negative allosteric NMDA receptor modulators

负变构NMDA受体调节剂的新型结合模式

Lotti, James S; Syrenne, Jed T; Benton, Avery J; Al-Mousawi, Ahmad; Cornelison, Lauren E; Trolinder, Christopher J; Yi, Feng; Zhang, Zhucheng; Yates-Hansen, Cindee K; McClelland, Levi J; Bosco, James; Rau, Andrew R; Clausen, Rasmus P; Hansen, Kasper B

Native architecture, allosteric modulation and gating mechanism of glycine-dependent NMDA receptors

甘氨酸依赖性NMDA受体的天然结构、变构调节和门控机制

Kim, Junhoe; Benton, Avery J; Lotti, James S; Rouzbeh, Nirvan; Hansen, Kasper B; Gouaux, Eric

The role of alpha-synuclein in synucleinopathy: Impact on lipid regulation at mitochondria-ER membranes.

α-突触核蛋白在突触核蛋白病中的作用:对线粒体-内质网膜脂质调节的影响

Barbuti Peter A, Guardia-Laguarta Cristina, Yun Taekyung, Chatila Zena K, Flowers Xena, Wong Chantel, Santos Bruno F R, Larsen Simone B, Lotti James S, Hattori Nobutaka, Bradshaw Elizabeth, Dettmer Ulf, Fanning Saranna, Menon Vilas, Reddy Hasini, Teich Andrew F, Krüger Rejko, Area-Gomez Estela, Przedborski Serge

Evaluation of allosteric N-methyl-d-aspartate receptor modulation by GluN2A-selective antagonists using pharmacological equilibrium modeling

利用药理平衡模型评估GluN2A选择性拮抗剂对N-甲基-D-天冬氨酸受体的变构调节作用

Lotti, James S; Jones, Jaron; Farnsworth, Jill C; Yi, Feng; Zhao, Fabao; Menniti, Frank S; Volkmann, Robert A; Clausen, Rasmus P; Hansen, Kasper B

Allosteric modulation of GluN1/GluN3 NMDA receptors by GluN1-selective competitive antagonists

GluN1选择性竞争性拮抗剂对GluN1/GluN3 NMDA受体的变构调节

Rouzbeh, Nirvan; Rau, Andrew R; Benton, Avery J; Yi, Feng; Anderson, Carly M; Johns, Mia R; Jensen, Loren; Lotti, James S; Holley, David C; Hansen, Kasper B

Discovery of (R)-2-amino-3-triazolpropanoic acid derivatives as NMDA receptor glycine site agonists with GluN2 subunit-specific activity

发现(R)-2-氨基-3-三唑丙酸衍生物作为NMDA受体甘氨酸位点激动剂,具有GluN2亚基特异性活性

Zhao, Fabao; Mazis, Georgios; Yi, Feng; Lotti, James S; Layeux, Michael S; Schultz, Eric P; Bunch, Lennart; Hansen, Kasper B; Clausen, Rasmus P