日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Optimization of Pyrazolo[3,4‑b]pyridine Analogues: Synthesis, In Vitro Anticancer Evaluation and In Vivo Pharmacokinetics

吡唑并[3,4-b]吡啶类似物的优化:合成、体外抗癌活性评价和体内药代动力学

Georgiou, Maria; Saxonis, Nikolaos; Palaiologou, Anastasia; Lampropoulou, Alexandra; Anagnostopoulos, Athanasios K; Pouli, Nicole; Marakos, Panagiotis; Lougiakis, Nikolaos; Tamvakopoulos, Constantin

Generation of a selective senolytic platform using a micelle-encapsulated Sudan Black B conjugated analog

利用胶束包裹的苏丹黑B偶联类似物构建选择性衰老细胞清除平台

Sophia Magkouta # ,Dimitris Veroutis # ,Angelos Papaspyropoulos # ,Maria Georgiou # ,Nikolaos Lougiakis ,Natassa Pippa ,Sophia Havaki ,Anastasia Palaiologou ,Dimitris-Foivos Thanos ,Konstantinos Kambas ,Nefeli Lagopati ,Nikos Boukos ,Nicole Pouli ,Panagiotis Marakos ,Athanassios Kotsinas ,Dimitris Thanos ,Konstantinos Evangelou ,Fotios Sampaziotis ,Constantin Tamvakopoulos ,Stergios Pispas ,Russell Petty ,Nicholas Kotopoulos ,Vassilis G Gorgoulis

Hit-to-Lead Optimization of Heterocyclic Carbonyloxycarboximidamides as Selective Antagonists at Human Adenosine A3 Receptor

杂环羰基氧甲酰亚胺作为人类腺苷 A3 受体选择性拮抗剂的命中到先导化合物优化

Xianglin Huang, Anna Chorianopoulou, Panagoula Kalkounou, Maria Georgiou, Athanasios Pousias, Amy Davies, Abigail Pearce, Matthew Harris, George Lambrinidis, Panagiotis Marakos, Nicole Pouli, Antonios Kolocouris, Nikolaos Lougiakis, Graham Ladds

One-step rapid tracking and isolation of senescent cells in cellular systems, tissues, or animal models via GLF16

通过 GLF16 一步快速追踪和分离细胞系统、组织或动物模型中的衰老细胞

Sophia Magkouta, Dimitris Veroutis, Athanasios Pousias, Angelos Papaspyropoulos, Kety Giannetti, Natassa Pippa, Nikolaos Lougiakis, Konstantinos Kambas, Nefeli Lagopati, Aikaterini Polyzou, Maria Georgiou, Maria Chountoulesi, Stergios Pispas, Spyros Foutadakis, Efthymios Kyrodimos, Nicole Pouli, Pan

A fluorophore-conjugated reagent enabling rapid detection, isolation and live tracking of senescent cells

一种荧光团结合试剂,可快速检测、分离和实时追踪衰老细胞

Sophia Magkouta, Dimitris Veroutis, Athanasios Pousias, Angelos Papaspyropoulos, Natassa Pippa, Nikolaos Lougiakis, Konstantinos Kambas, Nefeli Lagopati, Aikaterini Polyzou, Maria Georgiou, Maria Chountoulesi, Stergios Pispas, Spyros Foutadakis, Nicole Pouli, Panagiotis Marakos, Athanassios Kotsinas

SIRT2i_Predictor: A Machine Learning-Based Tool to Facilitate the Discovery of Novel SIRT2 Inhibitors

SIRT2i_Predictor:一种基于机器学习的工具,用于促进新型SIRT2抑制剂的发现

Djokovic, Nemanja; Rahnasto-Rilla, Minna; Lougiakis, Nikolaos; Lahtela-Kakkonen, Maija; Nikolic, Katarina

Discovery of a High Affinity Adenosine A(1)/A(3) Receptor Antagonist with a Novel 7-Amino-pyrazolo[3,4-d]pyridazine Scaffold

发现一种具有新型 7-氨基吡唑并[3,4-d]哒嗪骨架的高亲和力腺苷 A(1)/A(3) 受体拮抗剂

Suchankova, Anna; Stampelou, Margarita; Koutsouki, Klontiana; Pousias, Athanasios; Dhingra, Lakshiv; Barkan, Kerry; Pouli, Nicole; Marakos, Panagiotis; Tenta, Roxane; Kolocouris, Antonios; Lougiakis, Nikolaos; Ladds, Graham

Immunotherapy Combined with Metronomic Dosing: An Effective Approach for the Treatment of NSCLC

免疫疗法联合节拍给药:治疗非小细胞肺癌的有效方法

Skavatsou, Eleni; Semitekolou, Maria; Morianos, Ioannis; Karampelas, Theodoros; Lougiakis, Nikolaos; Xanthou, Georgina; Tamvakopoulos, Constantin

Screening of Heteroaromatic Scaffolds against Cystathionine Beta-Synthase Enables Identification of Substituted Pyrazolo[3,4-c]Pyridines as Potent and Selective Orthosteric Inhibitors

针对胱硫醚 β-合酶的杂芳族骨架筛选可鉴定取代的吡唑并 [3,4-c] 吡啶作为有效且选择性的正构抑制剂

Anna-Maria Fantel, Vassilios Myrianthopoulos, Anastasios Georgoulis, Nikolaos Lougiakis, Iliana Zantza, George Lamprinidis, Fiona Augsburger, Panagiotis Marakos, Constantinos E Vorgias, Csaba Szabo, Nicole Pouli, Andreas Papapetropoulos, Emmanuel Mikros

Design and Synthesis of New Substituted Pyrazolopyridines with Potent Antiproliferative Activity

设计并合成具有强效抗增殖活性的新型取代吡唑并吡啶类化合物

Giannouli, Vassiliki; Lougiakis, Nikolaos; Kostakis, Ioannis K; Pouli, Nicole; Marakos, Panagiotis; Skaltsounis, Alexios-Leandros; Horne, David A; Nam, Sangkil; Gioti, Katerina; Tenta, Roxane