日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Above-Filter Digestion Proteomics Reveals Drug Targets and Localizes Ligand Binding Site

滤膜上消化蛋白质组学揭示药物靶点并定位配体结合位点

Sokolova, Bohdana; Gharibi, Hassan; Jafari, Maryam; Lyu, Hezheng; Lovera, Silvia; Gaetani, Massimiliano; Saei, Amir Ata; Zubarev, Roman A

Elucidation of the mechanism of partial activation of EPAC1 allosteric modulators by Markov state modelling

利用马尔可夫状态模型阐明EPAC1变构调节剂部分激活的机制

Hardie, Adele; Powell, Frederick G; Lovera, Silvia; Yarwood, Stephen J; Barker, Graeme; Michel, Julien

Identification of a Lipid-Exposed Extrahelical Binding Site for Positive Allosteric Modulators of the Dopamine D(2) Receptor.

鉴定多巴胺 D(2) 受体正变构调节剂的脂质暴露螺旋外结合位点

Lim Herman D, Bartuzi Damian, Keen Alastair C, Rauffenbart Caroline, Glenn Jacqueline, Charlton Steven J, Lovera Silvia, Sands Zara A, Ates Ali, Wood Martyn, Canals Meritxell, Javitch Jonathan A, Carlsson Jens, Lane J Robert

Deconstructing allostery by computational assessment of the binding determinants of allosteric PTP1B modulators

通过计算评估变构PTP1B调节剂的结合决定因素来解构变构作用

Hardie, Adele; Cossins, Benjamin P; Lovera, Silvia; Michel, Julien

Crystal structure of dopamine D1 receptor in complex with G protein and a non-catechol agonist

多巴胺D1受体与G蛋白和非儿茶酚激动剂复合物的晶体结构

Sun, Bingfa; Feng, Dan; Chu, Matthew Ling-Hon; Fish, Inbar; Lovera, Silvia; Sands, Zara A; Kelm, Sebastian; Valade, Anne; Wood, Martyn; Ceska, Tom; Kobilka, Tong Sun; Lebon, Florence; Kobilka, Brian K

NaViA: a program for the visual analysis of complex mass spectra

NaViA:一款用于复杂质谱图可视化分析的程序

Quetschlich, Daniel; Esser, Tim K; Newport, Thomas D; Fiorentino, Francesco; Shutin, Denis; Chen, Siyun; Davis, Rachel; Lovera, Silvia; Liko, Idlir; Stansfeld, Phillip J; Robinson, Carol V

Reconstruction of apo A2A receptor activation pathways reveal ligand-competent intermediates and state-dependent cholesterol hotspots

重建载脂蛋白A2A受体激活通路揭示了配体结合的中间体和状态依赖性胆固醇热点

Lovera, Silvia; Cuzzolin, Alberto; Kelm, Sebastian; De Fabritiis, Gianni; Sands, Zara A