日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Anti-EGFR therapy can overcome acquired resistance to the third-generation ALK-tyrosine kinase inhibitor lorlatinib mediated by activation of EGFR.

抗 EGFR 疗法可以克服由 EGFR 激活介导的对第三代 ALK 酪氨酸激酶抑制剂劳拉替尼的获得性耐药性

Hu Chen, Lu Cong-Hua, Zheng Jie, Kang Jun, Huang Dai-Juan, He Chao, Liu Yi-Hui, Liu Zhan-Rui, Wu Di, Dou Yuan-Yao, Zhang Yi-Min, Lin Cai-Yu, Han Rui, He Yong

Brigatinib, a newly discovered AXL inhibitor, suppresses AXL-mediated acquired resistance to osimertinib in EGFR-mutated non-small cell lung cancer.

Brigatinib 是一种新发现的 AXL 抑制剂,可抑制 EGFR 突变型非小细胞肺癌中 AXL 介导的对奥希替尼的获得性耐药性

Han Rui, Lu Cong-Hua, Hu Chen, Dou Yuan-Yao, Kang Jun, Lin Cai-Yu, Wu Di, Jiang Wei-Ling, Yin Guo-Qing, He Yong