日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Quantitative live cell imaging of a tauopathy model enables the identification of a polypharmacological drug candidate that restores physiological microtubule interaction

tau 蛋白病模型的定量活细胞成像能够识别出可恢复生理微管相互作用的多药理学候选药物

Luca Pinzi #, Christian Conze #, Nicolo Bisi, Gabriele Dalla Torre, Ahmed Soliman, Nanci Monteiro-Abreu, Nataliya I Trushina, Andrea Krusenbaum, Maryam Khodaei Dolouei, Andrea Hellwig, Michael S Christodoulou, Daniele Passarella, Lidia Bakota, Giulio Rastelli, Roland Brandt

Searching for Novel HDAC6/Hsp90 Dual Inhibitors with Anti-Prostate Cancer Activity: In Silico Screening and In Vitro Evaluation

寻找具有抗前列腺癌活性的新型 HDAC6/Hsp90 双重抑制剂:计算机筛选和体外评估

Luca Pinzi, Silvia Belluti, Isabella Piccinini, Carol Imbriano, Giulio Rastelli

Antifungal Activity and DNA Topoisomerase Inhibition of Hydrolysable Tannins from Punica granatum L

石榴水解单宁的抗真菌活性和 DNA 拓扑异构酶抑制作用

Virginia Brighenti, Ramona Iseppi, Luca Pinzi, Annamaria Mincuzzi, Antonio Ippolito, Patrizia Messi, Simona Marianna Sanzani, Giulio Rastelli, Federica Pellati

Design of Dual Inhibitors of Histone Deacetylase 6 and Heat Shock Protein 90

组蛋白去乙酰化酶 6 和热休克蛋白 90 双重抑制剂的设计

Luca Pinzi, Rosaria Benedetti, Lucia Altucci, Giulio Rastelli