A Novel Small Molecule Allosteric Inhibitor of IL-17A from a DNA-Encoded Library
从DNA编码库中筛选出一种新型IL-17A小分子变构抑制剂
期刊:ACS Medicinal Chemistry Letters
影响因子:4
doi:10.1021/acsmedchemlett.5c00502
Milla, Marcos E; Blevitt, Jonathan M; Goldberg, Steven D; Armstrong, Anthony A; Blain, Katherine Y; Herman, Krystal L; Liu, Annie X; Luna, Rosa; Milligan, Cynthia M; Patrick, Aaron N; Steele, Ruth A; Bembenek, Scott D; Centrella, Paolo; Clark, Matthew A; Cuozzo, John W; Disch, Jeremy S; Domingo, Derrick; Hunt, Avery; Hupp, Christoper D; Keefe, Anthony D; Luo, Jinquan; Mirzadegan, Tara; Nelen, Marina I; Resnicow, Daniel I; Sigel, Eric A; Soutter, Holly H; Troast, Dawn M; Xue, Xiaohua; Yi, Fang; Zhang, Ying; Jackson, Paul F; Edwards, James P; Lumb, Kevin J