日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Assembling Ternary Dead-End Complex for Covalent Trapping of Protein Lysine Methyltransferases

组装三元死端复合物以共价捕获蛋白质赖氨酸甲基转移酶

Zong, Yu; Zhang, Nawei; Lin, Jason; Li, Zhizhong; Zou, Yuqiao; Chaudhuri, Rohit; Luo, Minkui

Discovery of a Potent, Selective, and In Vivo Efficacious Covalent Inhibitor for Lysine Methyltransferase SETD8

发现一种高效、选择性强且体内有效的赖氨酸甲基转移酶SETD8共价抑制剂

Chen, He; Dutta, Rudra Prasad; Li, Zhizhong; Zhong, Yue; Ma, Anqi; Park, Kwang-Su; Kottur, Jithesh; Park, Alison; Babault, Nicolas; Wang, Ke; Wang, Dandan; Xiong, Yan; Kaniskan, H Ümit; Luo, Minkui; Parekh, Samir; Jin, Jian

SGSS05-NS3, a covalent SETD8 inhibitor that activates p53 pathway in neuroblastoma

SGSS05-NS3 是一种共价 SETD8 抑制剂,可激活神经母细胞瘤中的 p53 通路。

Liu, Zhihui; Bagchi, Sukriti; Yan, Chunhua; Hu, Ying; Blum, Gil; Ma, Anqi; Jin, Jian; Luo, Minkui; Di Bella, Sebastiano; Verona, Francesco; Appella, Ettore; Giannini, Giuseppe; Thiele, Carol J; Veschi, Veronica

PRMT1-mediated metabolic reprogramming promotes leukemogenesis

PRMT1介导的代谢重编程促进白血病发生

Su, Hairui; Sun, Yong; Guo, Han; Sun, Chiao-Wang; Chen, Qiuying; Liu, Szumam; Li, Anlun; Gao, Min; Zhao, Rui; Raffel, Glen; Jin, Jian; Qu, Cheng-Kui; Yu, Michael; Klug, Christopher A; Zheng, George Y; Ballinger, Scott; Kutny, Matthew; Zheng, Long X; Chong, Zechen; Senevirathne, Chamara; Gross, Steven; Chen, Yabing; Luo, Minkui; Zhao, Xinyang

Crystal structure of SARS-CoV-2 nsp10-nsp16 in complex with small molecule inhibitors, SS148 and WZ16

SARS-CoV-2 nsp10-nsp16 与小分子抑制剂 SS148 和 WZ16 复合物的晶体结构

Klima, Martin; Khalili Yazdi, Aliakbar; Li, Fengling; Chau, Irene; Hajian, Taraneh; Bolotokova, Albina; Kaniskan, H Ümit; Han, Yulin; Wang, Ke; Li, Deyao; Luo, Minkui; Jin, Jian; Boura, Evzen; Vedadi, Masoud

Harnessing nanotechnology to expand the toolbox of chemical biology

利用纳米技术拓展化学生物学的工具箱

Williams, Ryan M; Chen, Shi; Langenbacher, Rachel E; Galassi, Thomas V; Harvey, Jackson D; Jena, Prakrit V; Budhathoki-Uprety, Januka; Luo, Minkui; Heller, Daniel A

Nanoreporter of an Enzymatic Suicide Inactivation Pathway

酶促自杀失活途径的纳米报告分子

Yaari, Zvi; Cheung, Justin M; Baker, Hanan A; Frederiksen, Rune S; Jena, Prakrit V; Horoszko, Christopher P; Jiao, Fang; Scheuring, Simon; Luo, Minkui; Heller, Daniel A

Correction: A chemical probe of CARM1 alters epigenetic plasticity against breast cancer cell invasion

更正:CARM1 的化学探针可改变表观遗传可塑性,从而抑制乳腺癌细胞侵袭

Cai, Xiao-Chuan; Zhang, Tuo; Kim, Eui-Jun; Jiang, Ming; Wang, Ke; Wang, Junyi; Chen, Shi; Zhang, Nawei; Wu, Hong; Li, Fengling; Dela Seña, Carlo C; Zeng, Hong; Vivcharuk, Victor; Niu, Xiang; Zheng, Weihong; Lee, Jonghan P; Chen, Yuling; Barsyte, Dalia; Szewczyk, Magda; Hajian, Taraneh; Ibáñez, Glorymar; Dong, Aiping; Dombrovski, Ludmila; Zhang, Zhenyu; Deng, Haiteng; Min, Jinrong; Arrowsmith, Cheryl H; Mazutis, Linas; Shi, Lei; Vedadi, Masoud; Brown, Peter J; Xiang, Jenny; Qin, Li-Xuan; Xu, Wei; Luo, Minkui

Chemical and Biochemical Perspectives of Protein Lysine Methylation

蛋白质赖氨酸甲基化的化学和生物化学视角

Luo, Minkui

N(6)-Allyladenosine: A New Small Molecule for RNA Labeling Identified by Mutation Assay

N(6)-烯丙基腺苷:一种通过突变分析鉴定的用于RNA标记的新型小分子

Shu, Xiao; Dai, Qing; Wu, Tong; Bothwell, Ian R; Yue, Yanan; Zhang, Zezhou; Cao, Jie; Fei, Qili; Luo, Minkui; He, Chuan; Liu, Jianzhao