日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Single-cell RNA sequencing reveals diverse B cell phenotypes in patients with anti-NMDAR encephalitis

单细胞 RNA 测序揭示抗 NMDAR 脑炎患者的 B 细胞表型多样

Sisi Li, Xiang Hu, Minjin Wang, Luoting Yu, Qi Zhang, Jing Xiao, Zhen Hong, Dong Zhou, Jinmei Li

Discovery of novel reversible inhibitor of DprE1 based on benzomorpholine for the treatment of tuberculosis

发现基于苯并吗啉的新型可逆性 DprE1 抑制剂用于治疗结核病

Wang Xiang #, Hualong He #, Xianjie Duan #, Zhiqun He, Xinyue Xu, Mengya Liao, Fei Teng, Xiao Li, Tianwen Luo, Jumei Zeng, Luoting Yu, Chao Gao

A novel VEGFR inhibitor ZLF-095 with potent antitumor activity and low toxicity

具有强抗肿瘤活性和低毒性的新型 VEGFR 抑制剂 ZLF-095

Xiao Li, Jia Wang, Qianqian Wang, Tianwen Luo, Xuejiao Song, Guoquan Wan, Zhanzhan Feng, Xiaojie He, Qian Lei, Ying Xu, Xinyu You, Luoting Yu, Lidan Zhang, Lifeng Zhao

Covalent inhibitors of EZH2: Design, synthesis and evaluation

EZH2 共价抑制剂:设计、合成与评价

Qiangsheng Zhang, Xinyi Chen, Xi Hu, Xianjie Duan, Guoquan Wan, Lu Li, Qiang Feng, Yiqian Zhang, Ningyu Wang, Luoting Yu

Nifuroxazide ameliorates pulmonary fibrosis by blocking myofibroblast genesis: a drug repurposing study

硝呋嗪通过抑制肌成纤维细胞生成改善肺纤维化:一项药物再利用研究

Cailing Gan # ,Qianyu Zhang # ,Hongyao Liu ,Guan Wang ,Liqun Wang ,Yali Li ,Zui Tan ,Wenya Yin ,Yuqin Yao ,Yongmei Xie ,Liang Ouyang ,Luoting Yu ,Tinghong Ye

A novel small molecule RK-019 inhibits FGFR2-amplification gastric cancer cell proliferation and induces apoptosis in vitro and in vivo

新型小分子RK-019抑制FGFR2扩增胃癌细胞增殖并在体内外诱导细胞凋亡

Jun Zeng, Kai Ran, Xinyue Li, Longyue Tao, Qiwei Wang, Jiangtao Ren, Rong Hu, Yongxia Zhu, Zhihao Liu, Luoting Yu

A novel multikinase inhibitor SKLB-YTH-60 ameliorates inflammation and fibrosis in bleomycin-induced lung fibrosis mouse models

新型多激酶抑制剂 SKLB-YTH-60 可改善博来霉素诱导的肺纤维化小鼠模型中的炎症和纤维化

Hongyao Liu, Xiuli Wu, Cailing Gan, Liqun Wang, Guan Wang, Lin Yue, Zhihao Liu, Wei Wei, Xingping Su, Qianyu Zhang, Zui Tan, Yuqin Yao, Liang Ouyang, Luoting Yu, Tinghong Ye

Synthesis and biological evaluation of indazole derivatives as anti-cancer agents

吲唑衍生物的合成及抗癌活性评价

Wei Wei, Zhihao Liu, Xiuli Wu, Cailing Gan, Xingping Su, Hongyao Liu, Hanyun Que, Qianyu Zhang, Qiang Xue, Lin Yue, Luoting Yu, Tinghong Ye

Preclinical evaluation of Amphihevir, a first-in-class clinical Hepatitis C virus NS4B inhibitor

首创临床丙型肝炎病毒 NS4B 抑制剂 Amphihevir 的临床前评估

Xin Tao, Ningyu Wang, Jianfei Wang, Zhifei Fu, Zhengxian Gu, Yang Zhang, Shuhui Chen, Lichun Wang, Luoting Yu

Corrigendum: Selective inhibition of EZH2 by ZLD1039 blocks H3K27methylation and leads to potent anti-tumor activity in breast cancer

更正:ZLD1039 选择性抑制 EZH2 可阻断 H3K27 甲基化,从而对乳腺癌产生强大的抗肿瘤活性

Xuejiao Song, Tiantao Gao, Ningyu Wang, Qiang Feng, Xinyu You, Tinghong Ye, Qian Lei, Yongxia Zhu, Menghua Xiong, Yong Xia, Fangfang Yang, Yaojie Shi, Yuquan Wei, Lidan Zhang, Luoting Yu