日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Special Issue "Biosynthesis and Application of Natural Compound"

特刊“天然化合物的生物合成与应用”

Luzina, Olga A; Volcho, Konstantin P

Usnic Acid Derivatives as Inhibitors of Mycobacterium tuberculosis Uracil-DNA Glycosylase

地衣酸衍生物作为结核分枝杆菌尿嘧啶-DNA糖苷酶抑制剂

Filimonov, Aleksandr S; Zateeva, Maria V; Mechetin, Grigory V; Luzina, Olga A; Eurtivong, Chatchakorn; Sari, Suat; Endutkin, Anton V; Reynisson, Jóhannes; Volcho, Konstantin P; Salakhutdinov, Nariman F; Zharkov, Dmitry O

The Influence of TDP1 Inhibitor Usnic Acid Derivative OL9-116 on the Effects of Topotecan in Human Cells

TDP1抑制剂乌斯尼酸衍生物OL9-116对拓扑替康在人细胞中作用的影响

Kornienko, Tatyana E; Chepanova, Arina A; Kolobenko, Maria V; Chernyshova, Irina A; Zakharenko, Alexandra L; Venzel, Artur S; Dyrkheeva, Nadezhda S; Markov, Andrey V; Anarbaev, Rashid O; Naumenko, Konstantin N; Luzina, Olga A; Salakhutdinov, Nariman F; Ivanisenko, Vladimir A; Lavrik, Olga I

Transcriptomic Analysis of TDP1-Knockout HEK293A Cells Treated with the TDP1 Inhibitor (Usnic Acid Derivative)

用TDP1抑制剂(乌斯尼酸衍生物)处理TDP1敲除HEK293A细胞的转录组分析

Zakharenko, Alexandra L; Dyrkheeva, Nadezhda S; Markov, Andrey V; Kleshchev, Maxim A; Ryabchikova, Elena I; Malakhova, Anastasia A; Orishchenko, Konstantin E; Okorokova, Larisa S; Shtokalo, Dmitriy N; Medvedev, Sergey P; Zakian, Suren M; Tupikin, Alexey A; Kabilov, Marsel R; Luzina, Olga A; Deyev, Sergey M; Lavrik, Olga I

Design and Biological Evaluation of Monoterpene-Conjugated (S)-2-Ethoxy-3-(4-(4-hydroxyphenethoxy)phenyl)propanoic Acids as New Dual PPARα/γ Agonists

单萜共轭物(S)-2-乙氧基-3-(4-(4-羟基苯乙氧基)苯基)丙酸作为新型双重PPARα/γ激动剂的设计与生物学评价

Borisov, Sergey A; Blokhin, Mikhail E; Meshkova, Yulia V; Marenina, Maria K; Zhukova, Nataliya A; Pavlova, Sophia V; Lastovka, Anastasiya V; Fomenko, Vladislav V; Zhurakovsky, Igor P; Luzina, Olga A; Khvostov, Mikhail V; Kudlay, Dmitry A; Salakhutdinov, Nariman F

Organoselenium compounds as an enriched source for the discovery of new antimicrobial agents.

有机硒化合物是发现新型抗菌剂的丰富来源

Friberg Louise I M, Kavanagh Angela, Amado Maite, Lowe Gabrielle, Zuegg Johannes, Novais de Paula Michelle, Onawole Abdulmujeeb, Floyd Holly E E, Kravchenko Angelina N, Guan Davy, Elliott Alysha G, Kuchar Julia, Mohr Fabian, Luzina Olga, Salakhutdinov Nariman, Volcho Konstantin, Farrukh Hafiz S U B, Kalsoom Umme, Saleem Rahman S Z, Blanchfield Joanne, Blaskovich Mark A T, Hansford Karl A

The Potential of Usnic-Acid-Based Thiazolo-Thiophenes as Inhibitors of the Main Protease of SARS-CoV-2 Viruses

基于地衣酸的噻唑并噻吩类化合物作为SARS-CoV-2病毒主蛋白酶抑制剂的潜力

Yarovaya, Olga I; Filimonov, Aleksandr S; Baev, Dmitriy S; Borisevich, Sophia S; Zaykovskaya, Anna V; Chirkova, Varvara Yu; Marenina, Mariya K; Meshkova, Yulia V; Belenkaya, Svetlana V; Shcherbakov, Dmitriy N; Gureev, Maxim A; Luzina, Olga A; Pyankov, Oleg V; Salakhutdinov, Nariman F; Khvostov, Mikhail V

Natural Products and Their Derivatives as Inhibitors of the DNA Repair Enzyme Tyrosyl-DNA Phosphodiesterase 1

天然产物及其衍生物作为DNA修复酶酪氨酰-DNA磷酸二酯酶1的抑制剂

Zakharenko, Alexandra L; Luzina, Olga A; Chepanova, Arina A; Dyrkheeva, Nadezhda S; Salakhutdinov, Nariman F; Lavrik, Olga I

Usnic Acid Derivatives Inhibit DNA Repair Enzymes Tyrosyl-DNA Phosphodiesterases 1 and 2 and Act as Potential Anticancer Agents

乌斯尼酸衍生物抑制DNA修复酶酪氨酰-DNA磷酸二酯酶1和2,并作为潜在的抗癌剂发挥作用。

Zakharenko, Alexandra L; Dyrkheeva, Nadezhda S; Luzina, Olga A; Filimonov, Aleksandr S; Mozhaitsev, Evgenii S; Malakhova, Anastasia A; Medvedev, Sergey P; Zakian, Suren M; Salakhutdinov, Nariman F; Lavrik, Olga I

Study of Hypoglycemic Activity of Novel 9-N-alkyltetrahydroberberine Derivatives

新型9-N-烷基四氢小檗碱衍生物降血糖活性的研究

Khvostov, Mikhail V; Gladkova, Elizaveta D; Borisov, Sergey A; Fedotova, Marina S; Zhukova, Nataliya A; Marenina, Mariya K; Meshkova, Yuliya V; Luzina, Olga A; Tolstikova, Tatiana G; Salakhutdinov, Nariman F