日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Development of PolyHis-Targeting PROTAC Degraders

开发针对多聚组氨酸的PROTAC降解剂

Chen, Hui; Zhu, Dong; Billitti, Monica; Sun, Annan; Jin, Lingtao; Moser, Emily; Mivechi, Nahid F; Zheng, Guangrong; Lv, Dongwen

Indomethacin exerts both cyclooxygenase inhibition-dependent and independent mechanisms to enhance chemo-immunotherapy in mice

吲哚美辛通过环氧合酶抑制依赖性和非依赖性机制增强小鼠的化疗免疫疗法。

Okoko, Ogacheko D; Aboelella, Nada S; Ye, Yan; Wang, Xin; Simon, Samson E; Gazi, Md Yeashin; Enriquez Castro, Victor J; Kehinde-Ige, Mercy; Brandle, Caitlin; Lv, Dongwen; Wolff, David W; Hedrick, Catherine C; Piazza, Gary; Shi, Huidong; Zhou, Gang

CD36-mediated endocytosis of proteolysis-targeting chimeras.

CD36介导的靶向蛋白水解嵌合体的内吞作用

Wang Zhengyu, Pan Bo-Syong, Manne Rajesh Kumar, Chen Jungang, Lv Dongwen, Wang Minmin, Tran Phuc, Weldemichael Tsigereda, Yan Wei, Zhou Hongfei, Martinez Gloria M, Shao Jingwei, Hsu Che-Chia, Hromas Robert, Zhou Daohong, Qin Zhiqiang, Lin Hui-Kuan, Li Hong-Yu

Discovery of Dual BCL-xL/BCL-w Degraders by Exploiting the Bis(sulfonyl)benzene Ring of ABT-263 as a Linkage Vector

利用ABT-263的双(磺酰基)苯环作为连接载体,发现双重BCL-xL/BCL-w降解剂

Poddar, Saikat K; Yang, Yang; Pal, Pratik; Jin, Zeng; Pei, Jing; Xiao, Yufeng; Hu, Wanyi; Zhang, Peiyi; Adekunbi, Praise; Thummuri, Dinesh; Yuan, Yaxia; Lv, Dongwen; Pelletier, J Peter R; Zhang, Weizhou; Zhou, Daohong; Zheng, Guangrong

Single-Assay Characterization of Ternary Complex Assembly and Activity in Targeted Protein Degradation.

单次检测表征靶向蛋白质降解中三元复合物的组装和活性

Yu Corey H, Dougherty Vi, Lv Dongwen, Ebadi Pirouz, Dubey Shikha, Nayak Digant, Nayak Anindita, Zhou Daohong, Olsen Shaun K, Ivanov Dmitri N

NSD2 drives t(4;14) myeloma cell dependence on adenylate kinase 2 by diverting one-carbon metabolism to the epigenome.

NSD2 通过将一碳代谢转移到表观基因组,驱动 t(4;14) 骨髓瘤细胞对腺苷酸激酶 2 的依赖性

Sobh Amin, Encinas Elena, Patel Alisha, Surapaneni Greeshma, Bonilla Emilie, Kaestner Charlotte, Poullard Janai, Clerio Monica, Vasan Karthik, Freeman Tzipporah, Lv Dongwen, Dupéré-Richer Daphné, Riva Alberto, Barwick Benjamin G, Zhou Daohong, Boise Lawrence H, Mitsiades Constantine S, Kim Baek, Bennett Richard L, Chandel Navdeep S, Licht Jonathan D

Bifunctional Peptide Nanofibrils for Targeted Protein Degradation

用于靶向蛋白质降解的双功能肽纳米纤维

Lin, Zongtao; Garcia, Benjamin A; Lv, Dongwen

Targeted Protein Degradation: Current and Emerging Approaches for E3 Ligase Deconvolution

靶向蛋白质降解:E3连接酶解卷积的当前和新兴方法

Xiao, Yufeng; Yuan, Yaxia; Liu, Yi; Lin, Zongtao; Zheng, Guangrong; Zhou, Daohong; Lv, Dongwen

Automation to Enable High-Throughput Chemical Proteomics

自动化助力高通量化学蛋白质组学

Lin, Zongtao; Gongora, Joanna; Liu, Xingyu; Xie, Yixuan; Zhao, Chenfeng; Lv, Dongwen; Garcia, Benjamin A

Proteolysis targeting chimeras (PROTACs) are emerging therapeutics for hematologic malignancies

蛋白水解靶向嵌合体(PROTACs)是治疗血液系统恶性肿瘤的新兴疗法。

He, Yonghan; Khan, Sajid; Huo, Zhiguang; Lv, Dongwen; Zhang, Xuan; Liu, Xingui; Yuan, Yaxia; Hromas, Robert; Xu, Mingjiang; Zheng, Guangrong; Zhou, Daohong