日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Deubiquitinase-targeting chimeras for targeted protein stabilization

去泛素化酶靶向嵌合体用于靶向蛋白质稳定

Nathaniel J Henning #, Lydia Boike #, Jessica N Spradlin, Carl C Ward, Gang Liu, Erika Zhang, Bridget P Belcher, Scott M Brittain, Matthew J Hesse, Dustin Dovala, Lynn M McGregor, Rachel Valdez Misiolek, Lindsey W Plasschaert, David J Rowlands, Feng Wang, Andreas O Frank, Daniel Fuller, Abigail R Es

Chemoproteomics-enabled discovery of covalent RNF114-based degraders that mimic natural product function

化学蛋白质组学助力发现可模拟天然产物功能的共价RNF114基降解剂

Mai Luo,Jessica N Spradlin,Lydia Boike,Bingqi Tong,Scott M Brittain,Jeffrey M McKenna,John A Tallarico,Markus Schirle,Thomas J Maimone,Daniel K Nomura

Discovery of a Functional Covalent Ligand Targeting an Intrinsically Disordered Cysteine within MYC

发现针对 MYC 内固有无序半胱氨酸的功能性共价配体

Lydia Boike, Alexander G Cioffi, Felix C Majewski, Jennifer Co, Nathaniel J Henning, Michael D Jones, Gang Liu, Jeffrey M McKenna, John A Tallarico, Markus Schirle, Daniel K Nomura