日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Newly Developed CK1-Specific Inhibitors Show Specifically Stronger Effects on CK1 Mutants and Colon Cancer Cell Lines

新开发的 CK1 特异性抑制剂对 CK1 突变体和结肠癌细胞系表现出更强的作用

Congxing Liu, Lydia Witt, Chiara Ianes, Joachim Bischof, Marie-Thérèse Bammert, Joana Baier, Stefan Kirschner, Doris Henne-Bruns, Pengfei Xu, Marko Kornmann, Christian Peifer, Uwe Knippschild

Optimized 4,5-Diarylimidazoles as Potent/Selective Inhibitors of Protein Kinase CK1δ and Their Structural Relation to p38α MAPK

优化的4,5-二芳基咪唑类化合物作为蛋白激酶CK1δ的强效/选择性抑制剂及其与p38α MAPK的结构关系

Jakob Halekotte,Lydia Witt,Chiara Ianes,Marc Krüger,Mike Bührmann,Daniel Rauh,Christian Pichlo,Elena Brunstein,Andreas Luxenburger,Ulrich Baumann,Uwe Knippschild,Joachim Bischof,Christian Peifer