日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Anti-Infective Properties, Cytotoxicity, and In Silico ADME Parameters of Novel 4'-(Piperazin-1-yl)benzanilides.

新型 4'-(哌嗪-1-基)苯甲酰化合物的抗感染特性、细胞毒性和计算机模拟 ADME 参数

Hermann Theresa, Harzl Sarah, Wallner Robin, Prettner Elke, Pferschy-Wenzig Eva-Maria, Cal Monica, Mäser Pascal, Weis Robert

Incomplete Plasmodium falciparum growth inhibition following piperaquine treatment translates into increased parasite viability in the in vitro parasite reduction ratio assay.

哌喹治疗后恶性疟原虫生长抑制不完全,导致体外寄生虫减少率试验中寄生虫存活率增加

Walz Annabelle, Sax Sibylle, Scheurer Christian, Tamasi Balint, Mäser Pascal, Wittlin Sergio

Studying Target-Engagement of Anti-Infectives by Solvent-Induced Protein Precipitation and Quantitative Mass Spectrometry.

利用溶剂诱导蛋白质沉淀和定量质谱法研究抗感染药物的靶向结合

Bizzarri Lorenzo, Steinbrunn Dominik, Quennesson Thibaut, Lacour Antoine, Bianchino Gabriella Ines, Bravo Patricia, Chaignon Philippe, Lohse Jonas, Mäser Pascal, Seemann Myriam, Calenbergh Serge Van, Hirsch Anna K H, Hahne Hannes

Integral Solvent-Induced Protein Precipitation for Target-Engagement Studies in Plasmodium falciparum.

利用溶剂诱导蛋白质沉淀法研究恶性疟原虫的靶标结合

Bravo Patricia, Bizzarri Lorenzo, Steinbrunn Dominik, Lohse Jonas, Hirsch Anna K H, Mäser Pascal, Rottmann Matthias, Hahne Hannes

New Derivatives of the Multi-Stage Active Malaria Box Compound MMV030666 and Their Antiplasmodial Potencies.

多阶段活性疟疾盒化合物 MMV030666 的新衍生物及其抗疟原虫效力

Hermann Theresa, Wallner Robin, Dolensky Johanna, Seebacher Werner, Pferschy-Wenzig Eva-Maria, Kaiser Marcel, Mäser Pascal, Weis Robert

2-(Nitroaryl)-5-Substituted-1,3,4-Thiadiazole Derivatives with Antiprotozoal Activities: In Vitro and In Vivo Study.

2-(硝基芳基)-5-取代-1,3,4-噻二唑衍生物的抗原生动物活性:体外和体内研究

Mousavi Alireza, Foroumadi Parham, Emamgholipour Zahra, Mäser Pascal, Kaiser Marcel, Foroumadi Alireza

Synthesis and Antiprotozoal Activity of Azabicyclo-Nonane Pyrimidine Hybrids.

氮杂双环壬烷嘧啶杂合物的合成及其抗原生动物活性

Hinteregger Clemens, Dolensky Johanna, Seebacher Werner, Saf Robert, Mäser Pascal, Kaiser Marcel, Weis Robert

Antiprotozoal Activity of Azabicyclo-Nonanes Linked to Tetrazole or Sulfonamide Cores.

与四唑或磺酰胺核心连接的氮杂双环壬烷的抗原生动物活性

Dolensky Johanna, Hinteregger Clemens, Leitner Andreas, Seebacher Werner, Saf Robert, Belaj Ferdinand, Mäser Pascal, Kaiser Marcel, Weis Robert

The 3-phosphoinositide-dependent protein kinase 1 is an essential upstream activator of protein kinase A in malaria parasites.

3-磷酸肌醇依赖性蛋白激酶 1 是疟原虫中蛋白激酶 A 的重要上游激活因子

Hitz Eva, Wiedemar Natalie, Passecker Armin, Graça Beatriz A S, Scheurer Christian, Wittlin Sergio, Brancucci Nicolas M B, Vakonakis Ioannis, Mäser Pascal, Voss Till S

New Acyl Derivatives of 3-Aminofurazanes and Their Antiplasmodial Activities.

3-氨基呋喃烷的新型酰基衍生物及其抗疟活性

Hermann Theresa, Hochegger Patrick, Dolensky Johanna, Seebacher Werner, Saf Robert, Kaiser Marcel, Mäser Pascal, Weis Robert