日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

PI3Kα Inhibitor and Degrader Inavolisib Can Co-opt FGFR2 to Enhance Responses in Patients with PIK3CA-Mutated Solid Tumors and in Preclinical Models.

PI3Kα抑制剂和降解剂Inavolisib可利用FGFR2增强PIK3CA突变实体瘤患者和临床前模型的疗效。

Juric Dejan, Song Kyung, Johnson Radia M, Accordino Melissa K, Bedard Philippe L, Cervantes Andrés, Gambardella Valentina, Hamilton Erika, Italiano Antoine, Kalinsky Kevin, Krop Ian E, Oliveira Mafalda, Saura Cristina, Schmid Peter, Turner Nicholas C, Varga Andreea, Gendreau Steven, Hwang Michael S, Kuang Zheng, Lau Jeffrey T, Lin Eva, Pham Trang, Maddalo Danilo, Rees Matthew G, Ronan Melissa M, Roth Jennifer A, Martin Scott, Sodir Nicole M, Sokol Ethan S, Whitfield Zachary J, Wong Alice, Yauch Robert L, Aimi Junko, Cheeti Sravanthi, Fredrickson Jill, Hilz Stephanie, Hafner Marc, Hutchinson Katherine E, Jin Yanling, Peters Ubong, Zingg Daniel, Royer-Joo Stephanie, Shankar Noopur, Schutzman Jennifer L, Jhaveri Komal L, Dey Anwesha

Nontargeted screening identifies mixtures of environmental pollutants that are associated with perturbations to amino acid and fatty acid metabolic pathways during early pregnancy

非靶向筛查可识别与早期妊娠期间氨基酸和脂肪酸代谢途径紊乱相关的环境污染物混合物。

Pedersen, Adam F; Petrick, Lauren M; Roth, Katherine; Yang, Zhao; Sitarik, Alexandra R; Maroli, Amith; Dolios, Georgia; Carignan, Courtney; Goodrich, Jaclyn M; Kerver, Jean M; Petriello, Michael

Engineering bioinspired, high-density collagen microgels with tunable intrafibrillar mineralization for accelerated osteogenesis in vitro and bone regeneration in vivo

构建仿生高密度胶原微凝胶,其纤维内矿化程度可调,可加速体外成骨和体内骨再生。

Vignolo, Sofia M; Roth, Daniela M; Fraga, May A A; Wu, Lillian; Cosgrove, Jameson A; Athirasala, Avathamsa; Lin, Angela S P; Guldberg, Robert E; Bertassoni, Luiz E

Synthesis and Biological Evaluation of Colibactin Derivatives

大肠杆菌素衍生物的合成及生物学评价

Airan, Yougant; Fedorova, Olga; Heer, Collin; Rees, Matthew G; Ronan, Melissa M; Roth, Jennifer A; Bindra, Ranjit S; Herzon, Seth B

Pregnancy- and age-associated variation in serum dehydroepiandrosterone concentrations in black and white rhinoceroses

黑犀牛和白犀牛血清脱氢表雄酮浓度的妊娠和年龄相关变化

Arbogast, Drew M; Metrione, Lara C; Jones, Marieke K; Donelan, Elizabeth M; Roth, Terri L; Freeman, Elizabeth W; Rispoli, Louisa A

Double plate fixation improves stiffness in a comminuted canine scapula fracture gap model compared to single plate fixation

与单钢板固定相比,双钢板固定可提高犬肩胛骨粉碎性骨折间隙模型的刚度。

Barrett, Faolain M; Roth, Josh D; Feller, Herman; McCarthy, Jessica

KDM4C inhibition blocks tumor growth in basal breast cancer by promoting cathepsin L-mediated histone H3 cleavage.

KDM4C 抑制剂通过促进组织蛋白酶 L 介导的组蛋白 H3 裂解来阻断基底型乳腺癌的肿瘤生长

Li Zheqi, Peluffo Guillermo, Stevens Laura E, Qiu Xintao, Seehawer Marco, Tawawalla Amatullah, Huang Xiao-Yun, Egri Shawn B, Raval Shaunak, McFadden Maeve, D'Santos Clive S, Papachristou Eva, Kingston Natalie L, Nishida Jun, Evans Kyle E, Seo Ji-Heui, Clement Kendell, Temko Daniel, Ekram Muhammad, Li Rong, Rees Matthew G, Ronan Melissa M, Roth Jennifer A, Simeonov Anton, Kales Stephen C, Rai Ganesha, Lal-Nag Madhu, Maloney David J, Jadhav Ajit, Michor Franziska, Meissner Alex, Balko Justin M, Carroll Jason S, Freedman Matthew L, Jaffe Jacob D, Papanastasiou Malvina, Long Henry W, Polyak Kornelia

Identification of a Selective Anticancer Agent from a Collection of Complex-And-Diverse Compounds Synthesized from Stevioside

从甜菊苷合成的一系列复杂多样的化合物中鉴定出一种选择性抗癌剂

Schaaf, Rachel E; Quirke, Jonathan C K; Ghavami, Maryam; Tonogai, Emily J; Lee, Hyang Yeon; Barlock, Samantha L; Trzupek, Thomas R; Abo, Kyle R; Rees, Matthew G; Ronan, Melissa M; Roth, Jennifer A; Hergenrother, Paul J

An allele-agnostic mutant-KRAS inhibitor suppresses tumor maintenance signals and reprograms tumor immunity in pancreatic cancer

一种不依赖于特定等位基因的突变型KRAS抑制剂可抑制肿瘤维持信号并重编程胰腺癌的肿瘤免疫。

McAndrews, Kathleen M; Paradiso, Francesca; Stalnecker, Clint A; Chellakkan, Benson S; Thege, Fredrik I; Peng, David H; Moreno Diaz, Barbara A; Sugimoto, Hikaru; Patel, Sarah I; Mahadevan, Krishnan K; Kirtley, Michelle L; Wills, Danielle; Sockwell, Amari M; Fonseca, Andre Luis F; Liu, Yunhe; Rajapakshe, Kimal I; Yee, Nathaniel G; Tran, Phuong Thao; Omar, Huda Alchikh; Tedeschi, Antonio; Schischlik-Siegl, Fiorella; Boghossian, Andrew S; Rees, Matthew G; Ronan, Melissa M; Roth, Jennifer A; Rudolph, Dorothea; Aichinger, Martin; Ebner, Florian; Artemov, Artem V; Lipp, Jesse; Pisarsky, Laura; Herrmann, Valerie Laura; Park, John; Rippmann, Jörg F; Schaaf, Otmar; Chandler, Vanessa; Williams, Mariah; Deckard, Charles E; Wang, Linghua; Der, Channing J; Vellano, Christopher; Guerrero, Paola A; Heffernan, Timothy P; Kalluri, Raghu; Maitra, Anirban

Tegavivint triggers TECR-dependent nonapoptotic cancer cell death

Tegavivint 诱导 TECR 依赖性非凋亡性癌细胞死亡

Leak, Logan; Wang, Ziwei; Joseph, Alby J; Johnson, Brianna; Chan, Alyssa A; Decosto, Cassandra M; Magtanong, Leslie; Ko, Pin-Joe; Lee, Weaverly Colleen; Ritho, Joan; Manukian, Sophia; Millner, Alec; Chitkara, Shweta; Salinas, Jennifer J; Skouta, Rachid; Rees, Matthew G; Ronan, Melissa M; Roth, Jennifer A; Myers, Chad L; Moffat, Jason; Boone, Charles; Bensinger, Steven J; Nathanson, David A; Atilla-Gokcumen, G Ekin; Moding, Everett J; Dixon, Scott J