日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Novel Triazoloquinoxaline-Based Tubulin Polymerization Inhibitor Induces Necroptosis and Significantly Inhibits Metastatic Melanoma Tumor Growth

一种新型三唑喹喔啉类微管蛋白聚合抑制剂可诱导坏死性凋亡并显著抑制转移性黑色素瘤肿瘤生长

Clark, Christopher J; Waddell, Shelby N; Tessmer, Garrett E; Womack, Carl B; Xie, Yang; Williams, Brittney D; Endraws, Meirola A; Huddleston, Cole T; Pulis, Keiluhn D; Thammathong, Joshua; Tanas, Kamil; Jangir, Beari A; Ma, Dejian; Bicker, Kevin L; Wang, Yaohong; Weissmiller, April M; Li, Wei; Banerjee, Souvik

Development of highly potent EP2 antagonists as novel anti-inflammatory neuroprotectants

开发高效EP2拮抗剂作为新型抗炎神经保护剂

Jiang, Chenyao; Cho, Eun Bee; Jin, Zhen; Bahraminejad, Sina; Ma, Dejian; Yu, Ying; Liu, Jiawang; Jiang, Jianxiong

Discovery of highly potent naphthalene/quinoline-based PAD inhibitors: Structure-activity relationship, selectivity, and cytotoxicity

高效萘/喹啉类PAD抑制剂的发现:构效关系、选择性和细胞毒性

Jia, Yijiang; Bahraminejad, Sina; Duan, Xin; Kong, Sydney; Taledaohan, Ayijiang; Jiang, Chenyao; Ma, Dejian; Jiang, Jianxiong; Wang, Yuji; Liu, Jiawang

Design and synthesis of novel 4-aryl-2-benzoyl-imidazoles as colchicine binding site inhibitors.

设计和合成新型 4-芳基-2-苯甲酰基咪唑类化合物作为秋水仙碱结合位点抑制剂

Albadari Najah, Xie Yang, Wang Qinghui, Miller Darcie J, Gruntz Judith Quadrozzi, Oldham Michael L, Chen Hao, Ma Dejian, Wu Zhongzhi, Miller Duane D, Li Wei

Extracellular Vesicle-Liposome-Darunavir Formulation for the Treatment of HIV Neuropathogenesis.

用于治疗 HIV 神经病变的细胞外囊泡-脂质体-达芦那韦制剂

Zhou Lina, Godse Sandip, Sinha Namita, Ma Dejian, Mirzahosseini Golnoush, Salman Mohd, Pulliam Paul, Tan Chalet, Singh Udai P, Ishrat Tauheed, Kochat Harry, Kumar Santosh

New structural scaffolds to enhance the metabolic stability of arginine-derived PAD4 inhibitors

新型结构支架增强精氨酸衍生的PAD4抑制剂的代谢稳定性

Jia, Yijiang; Bahraminejad, Sina; Jiang, Chenyao; Taledaohan, Ayijiang; Ma, Dejian; Jiang, Jianxiong; Wang, Yuji; Liu, Jiawang

Design and Crushing Behaviors Investigations of Novel High-Performance Bi-Tubular Tubes with Mixed Multicellular Configurations

新型高性能双管混合多胞结构的设计与压溃行为研究

Li, Zhaoji; Wang, Zhiwen; Ma, Dejian; Zeng, Qingliang; Ruan, Dong

Discovery of a potent and selective TRPC3 antagonist with neuroprotective effects.

发现了一种具有神经保护作用的强效选择性 TRPC3 拮抗剂

Wang Jiaxing, Zhang Sicheng, Boda Vijay K, Chen Hao, Park Hyunseo, Parmar Keyur, Ma Dejian, Miller Duane D, Meibohm Bernd, Du Jianyang, Liao Francesca-Fang, Wu Zhongzhi, Li Wei

Biological activity of a stable 6-aryl-2-benzoyl-pyridine colchicine-binding site inhibitor, 60c, in metastatic, triple-negative breast cancer.

稳定的 6-芳基-2-苯甲酰基-吡啶秋水仙碱结合位点抑制剂 60c 在转移性三阴性乳腺癌中的生物活性

Oluwalana Damilola, Adeleye Kelli L, Krutilina Raisa I, Chen Hao, Playa Hilaire, Deng Shanshan, Parke Deanna N, Abernathy John, Middleton Leona, Cullom Alexandra, Thalluri Bhargavi, Ma Dejian, Meibohm Bernd, Miller Duane D, Seagroves Tiffany N, Li Wei

Inhibiting De Novo Biosynthesis of Ceramide by L-Cycloserine Can Prevent Light-Induced Retinal Degeneration in Albino BALB/c Mice

L-环丝氨酸抑制神经酰胺从头合成可预防白化BALB/c小鼠的光诱导视网膜变性

Tahia, Faiza; Ma, Dejian; Stephenson, Daniel J; Basu, Sandip K; Del Mar, Nobel A; Lenchik, Nataliya; Kochat, Harry; Brown, Kennard; Chalfant, Charles E; Mandal, Nawajes