日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Defining substrate specificities of human RNA capping methyltransferases through quantitative assessment of independent yet cooperative activities.

通过对独立但协同活性的定量评估,确定人类 RNA 加帽甲基转移酶的底物特异性。

Taherian Fatemeh, Mabanglo Mark F, Hajian Taraneh, Tucker Sarah, Kalinic Emilija, Perveen Sumera, Aman Ahmed, Vedadi Masoud

Crystal structures of DCAF1-PROTAC-WDR5 ternary complexes provide insight into DCAF1 substrate specificity

DCAF1-PROTAC-WDR5三元复合物的晶体结构揭示了DCAF1的底物特异性

Mark F Mabanglo # ,Brian Wilson # ,Mahmoud Noureldin # ,Serah W Kimani ,Ahmed Mamai ,Chiara Krausser ,Héctor González-Álvarez ,Smriti Srivastava ,Mohammed Mohammed ,Laurent Hoffer ,Manuel Chan ,Jamie Avrumutsoae ,Alice Shi Ming Li ,Taraneh Hajian ,Sarah Tucker ,Stuart Green ,Magdalena Szewczyk ,Dalia Barsyte-Lovejoy ,Vijayaratnam Santhakumar ,Suzanne Ackloo ,Peter Loppnau ,Yanjun Li ,Almagul Seitova ,Taira Kiyota ,Jue George Wang ,Gilbert G Privé ,Douglas A Kuntz ,Bhashant Patel ,Vaibhavi Rathod ,Anand Vala ,Bhimsen Rout ,Ahmed Aman ,Gennady Poda ,David Uehling ,Jailall Ramnauth ,Levon Halabelian ,Richard Marcellus ,Rima Al-Awar ,Masoud Vedadi

Potent ClpP agonists with anticancer properties bind with improved structural complementarity and alter the mitochondrial N-terminome

具有抗癌特性的强效 ClpP 激动剂与改进的结构互补性结合并改变线粒体的 N 端

Mark F Mabanglo, Keith S Wong, Marim M Barghash, Elisa Leung, Stephanie H W Chuang, Afshan Ardalan, Emily M Majaesic, Cassandra J Wong, Shen Zhang, Henk Lang, Donald S Karanewsky, Andrew A Iwanowicz, Lee M Graves, Edwin J Iwanowicz, Anne-Claude Gingras, Walid A Houry

Recent structural insights into the mechanism of ClpP protease regulation by AAA+ chaperones and small molecules

近期对 AAA+ 分子伴侣和小分子调控 ClpP 蛋白酶机制的结构性研究进展

Mabanglo, Mark F; Houry, Walid A

Development of Antibiotics That Dysregulate the Neisserial ClpP Protease

开发能扰乱奈瑟菌ClpP蛋白酶活性的抗生素

Binepal, Gursonika; Mabanglo, Mark F; Goodreid, Jordan D; Leung, Elisa; Barghash, Marim M; Wong, Keith S; Lin, Funing; Cossette, Michele; Bansagi, Jazmin; Song, Boxi; Balasco Serrão, Vitor Hugo; Pai, Emil F; Batey, Robert A; Gray-Owen, Scott D; Houry, Walid A

Mitochondrial ClpP-Mediated Proteolysis Induces Selective Cancer Cell Lethality

线粒体 ClpP 介导的蛋白水解诱导选择性癌细胞致死

Jo Ishizawa, Sarah F Zarabi, R Eric Davis, Ondrej Halgas, Takenobu Nii, Yulia Jitkova, Ran Zhao, Jonathan St-Germain, Lauren E Heese, Grace Egan, Vivian R Ruvolo, Samir H Barghout, Yuki Nishida, Rose Hurren, Wencai Ma, Marcela Gronda, Todd Link, Keith Wong, Mark Mabanglo, Kensuke Kojima, Gautam Bort

ClpP protease activation results from the reorganization of the electrostatic interaction networks at the entrance pores.

ClpP 蛋白酶的激活是由于入口孔处静电相互作用网络的重组所致

Mabanglo Mark F, Leung Elisa, Vahidi Siavash, Seraphim Thiago V, Eger Bryan T, Bryson Steve, Bhandari Vaibhav, Zhou Jin Lin, Mao Yu-Qian, Rizzolo Kamran, Barghash Marim M, Goodreid Jordan D, Phanse Sadhna, Babu Mohan, Barbosa Leandro R S, Ramos Carlos H I, Batey Robert A, Kay Lewis E, Pai Emil F, Houry Walid A

Crystal structures of the fungal pathogen Aspergillus fumigatus protein farnesyltransferase complexed with substrates and inhibitors reveal features for antifungal drug design

真菌病原体烟曲霉蛋白法呢基转移酶与底物和抑制剂复合的晶体结构揭示了抗真菌药物设计的特征

Mark F Mabanglo, Michael A Hast, Nathan B Lubock, Homme W Hellinga, Lorena S Beese

Mutagenesis of isopentenyl phosphate kinase to enhance geranyl phosphate kinase activity

通过异戊烯基磷酸激酶诱变增强香叶基磷酸激酶活性

Mabanglo, Mark F; Pan, Jian-Jung; Shakya, Binita; Poulter, C Dale

X-ray structures of isopentenyl phosphate kinase

异戊烯基磷酸激酶的X射线晶体结构

Mabanglo, Mark F; Schubert, Heidi L; Chen, Mo; Hill, Christopher P; Poulter, C Dale