Discovery of VU6005649, a CNS Penetrant mGlu7/8 Receptor PAM Derived from a Series of Pyrazolo[1,5- a]pyrimidines
发现 VU6005649,一种源自一系列吡唑并[1,5- a]嘧啶的中枢神经系统渗透性 mGlu7/8 受体 PAM
期刊:ACS Medicinal Chemistry Letters
影响因子:3.5
doi:10.1021/acsmedchemlett.7b00317
Masahito Abe, Mabel Seto, Rocco G Gogliotti, Matthew T Loch, Katrina A Bollinger, Sichen Chang, Eileen M Engelberg, Vincent B Luscombe, Joel M Harp, Michael Bubser, Darren W Engers, Carrie K Jones, Alice L Rodriguez, Anna L Blobaum, P Jeffrey Conn, Colleen M Niswender, Craig W Lindsley