日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Deregulation of FOXF1/FENDRR from t(14;16)(q32;q24) defines a subtype of high-risk lineage ambiguous leukemia

t(14;16)(q32;q24)导致的FOXF1/FENDRR基因失调定义了一种高危谱系模糊白血病亚型。

Di Giacomo, Danika; Pölönen, Petri; Bardelli, Valentina; Kimura, Shunsuke; Pierini, Valentina; Pagliaro, Luca; Arniani, Silvia; Chang, Yunchao; Gao, Qingsong; Montefiori, Lindsey E; Wu, Yiming; Park, Chun Shik; Wright, William C; Vento, Federica; Wei, Huimei; Matteucci, Caterina; Lei, Shaohua; Rosikiewicz, Wojciech; Nardelli, Carlotta; Lema Fernandez, Anair Graciela; Østergaard, Anna; Backhaus, Emily A; Baviskar, Pradyumna; Cerrano, Marco; Leoncin, Matteo; Manabe, Atsushi; Hirabayashi, Shinsuke; Takita, Junko; Hasegawa, Daisuke; Miyamoto, Satoshi; Macchiarulo, Antonio; Xu, Jason; Teachey, David Trent; Roti, Giovanni; Iacobucci, Ilaria; La Starza, Roberta; Mecucci, Cristina; Mullighan, Charles G

Synthesis and structure-activity relationship study of a library of 1-substituted [1,2,4]triazolo[4,3-a]quinolines as valuable chemical probes for paraxonase-2 (PON2)

合成及构效关系研究1-取代[1,2,4]三唑并[4,3-a]喹啉类化合物库作为对对氧磷酶-2 (PON2) 有价值的化学探针

Bianconi, Elisa; Lampitella, Eros Antonio; Nigro, Fatima; Rossi, Ludovica; Zambri, Federico; Fava, Simone; Marone, Maria; Porzio, Elena; Macchiarulo, Antonio; Manco, Giuseppe; Marinozzi, Maura

Ligand-induced conformations and dynamic allosteric motions of IDO1 affecting the recruitment of a protein signaling partner.

配体诱导的 IDO1 构象和动态变构运动影响蛋白质信号伴侣的募集

Coletti Alice, Bianconi Elisa, Rossini Sofia, Altomare Alessandra, Butticè Andrea, Mazzoletti Daniele, Mondanelli Giada, Carotti Andrea, Aldini Giancarlo, Miggiano Riccardo, Orabona Ciriana, Salafsky Joshua, Macchiarulo Antonio

Adverse pro-tumorigenic effects of IDO1 catalytic inhibitors mediated by the non-enzymatic function of IDO1 in tumor cells

IDO1催化抑制剂通过IDO1在肿瘤细胞中的非酶促功能发挥促肿瘤作用

Rossini, Sofia; Ambrosino, Sara; Volpi, Claudia; Suvieri, Chiara; Pallotta, Maria Teresa; Belladonna, Maria Laura; Sorcini, Daniele; Macchiarulo, Antonio; Hennes, Elisabeth; Ziegler, Slava; Waldmann, Herbert; Orabona, Ciriana

Design, Synthesis, and Biological Characterization of Macromolecular Ester Prodrugs of a Selective Cyclooxygenase-2 Inhibitor

选择性环氧合酶-2抑制剂大分子酯前药的设计、合成和生物学表征

Saletti, Mario; Paolino, Marco; Venditti, Jacopo; Giuliani, Germano; Rossi, Antonietta; D'Avino, Danilo; Perna, Sara; Varfaj, Ina; Sardella, Roccaldo; Macchiarulo, Antonio; Maramai, Samuele; Lamponi, Stefania; Cappelli, Andrea; Anzini, Maurizio

Integrating post-event very high resolution SAR imagery and machine learning for building-level earthquake damage assessment

结合震后超高分辨率SAR图像和机器学习技术进行建筑物级地震破坏评估

Macchiarulo, Valentina; Giardina, Giorgia; Milillo, Pietro; Aktas, Yasemin D; Whitworth, Michael R Z

Epacadostat stabilizes the apo-form of IDO1 and signals a pro-tumorigenic pathway in human ovarian cancer cells

Epacadostat 可稳定 IDO1 的脱辅基形式,并在人类卵巢癌细胞中发出促肿瘤发生途径的信号

Sofia Rossini, Sara Ambrosino, Claudia Volpi, Maria Laura Belladonna, Maria Teresa Pallotta, Eleonora Panfili, Chiara Suvieri, Antonio Macchiarulo, Giada Mondanelli, Ciriana Orabona

A microbially produced AhR ligand promotes a Tph1-driven tolerogenic program in multiple sclerosis

微生物产生的 AhR 配体促进多发性硬化症中 Tph1 驱动的耐受性程序

Teresa Zelante, Giuseppe Paolicelli, Francesca Fallarino, Marco Gargaro, Gianluca Vascelli, Marco De Zuani, Jan Fric, Petra Laznickova, Marcela Hortova Kohoutkova, Antonio Macchiarulo, Daniela Dolciami, Giuseppe Pieraccini, Lorenzo Gaetani, Giulia Scalisi, Caterina Trevisan, Barbara Frossi, Carlo Pu

Identification of a Compound Inhibiting Both the Enzymatic and Nonenzymatic Functions of Indoleamine 2,3-Dioxygenase 1.

鉴定一种抑制吲哚胺 2,3-双加氧酶 1 的酶促和非酶促功能的化合物

Panfili Eleonora, Rezzi Sarah Jane, Adamo Annalisa, Mazzoletti Daniele, Massarotti Alberto, Miggiano Riccardo, Fallarini Silvia, Ambrosino Sara, Coletti Alice, Molinaro Pasquale, Milella Michele, Paiella Salvatore, Macchiarulo Antonio, Ugel Stefano, Pirali Tracey, Pallotta Maria Teresa

Achievable resolution for scalable Waveform Digitizing PET readout and comparison with ideal TDC-based readout with an application of DNN to optimal estimation including DOI

可扩展波形数字化PET读出可实现的分辨率,并与基于TDC的理想读出进行比较,应用DNN进行最优估计,包括DOI。

Macchiarulo, L; Chock, C; Mostafanezhad, I; Sabet, H