日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Deregulation of FOXF1/FENDRR from t(14;16)(q32;q24) defines a subtype of high-risk lineage ambiguous leukemia

t(14;16)(q32;q24)导致的FOXF1/FENDRR基因失调定义了一种高危谱系模糊白血病亚型。

Di Giacomo, Danika; Pölönen, Petri; Bardelli, Valentina; Kimura, Shunsuke; Pierini, Valentina; Pagliaro, Luca; Arniani, Silvia; Chang, Yunchao; Gao, Qingsong; Montefiori, Lindsey E; Wu, Yiming; Park, Chun Shik; Wright, William C; Vento, Federica; Wei, Huimei; Matteucci, Caterina; Lei, Shaohua; Rosikiewicz, Wojciech; Nardelli, Carlotta; Lema Fernandez, Anair Graciela; Østergaard, Anna; Backhaus, Emily A; Baviskar, Pradyumna; Cerrano, Marco; Leoncin, Matteo; Manabe, Atsushi; Hirabayashi, Shinsuke; Takita, Junko; Hasegawa, Daisuke; Miyamoto, Satoshi; Macchiarulo, Antonio; Xu, Jason; Teachey, David Trent; Roti, Giovanni; Iacobucci, Ilaria; La Starza, Roberta; Mecucci, Cristina; Mullighan, Charles G

Synthesis and structure-activity relationship study of a library of 1-substituted [1,2,4]triazolo[4,3-a]quinolines as valuable chemical probes for paraxonase-2 (PON2)

合成及构效关系研究1-取代[1,2,4]三唑并[4,3-a]喹啉类化合物库作为对对氧磷酶-2 (PON2) 有价值的化学探针

Bianconi, Elisa; Lampitella, Eros Antonio; Nigro, Fatima; Rossi, Ludovica; Zambri, Federico; Fava, Simone; Marone, Maria; Porzio, Elena; Macchiarulo, Antonio; Manco, Giuseppe; Marinozzi, Maura

Ligand-induced conformations and dynamic allosteric motions of IDO1 affecting the recruitment of a protein signaling partner.

配体诱导的 IDO1 构象和动态变构运动影响蛋白质信号伴侣的募集

Coletti Alice, Bianconi Elisa, Rossini Sofia, Altomare Alessandra, Butticè Andrea, Mazzoletti Daniele, Mondanelli Giada, Carotti Andrea, Aldini Giancarlo, Miggiano Riccardo, Orabona Ciriana, Salafsky Joshua, Macchiarulo Antonio

Adverse pro-tumorigenic effects of IDO1 catalytic inhibitors mediated by the non-enzymatic function of IDO1 in tumor cells

IDO1催化抑制剂通过IDO1在肿瘤细胞中的非酶促功能发挥促肿瘤作用

Rossini, Sofia; Ambrosino, Sara; Volpi, Claudia; Suvieri, Chiara; Pallotta, Maria Teresa; Belladonna, Maria Laura; Sorcini, Daniele; Macchiarulo, Antonio; Hennes, Elisabeth; Ziegler, Slava; Waldmann, Herbert; Orabona, Ciriana

Design, Synthesis, and Biological Characterization of Macromolecular Ester Prodrugs of a Selective Cyclooxygenase-2 Inhibitor

选择性环氧合酶-2抑制剂大分子酯前药的设计、合成和生物学表征

Saletti, Mario; Paolino, Marco; Venditti, Jacopo; Giuliani, Germano; Rossi, Antonietta; D'Avino, Danilo; Perna, Sara; Varfaj, Ina; Sardella, Roccaldo; Macchiarulo, Antonio; Maramai, Samuele; Lamponi, Stefania; Cappelli, Andrea; Anzini, Maurizio

Identification of a Compound Inhibiting Both the Enzymatic and Nonenzymatic Functions of Indoleamine 2,3-Dioxygenase 1.

鉴定一种抑制吲哚胺 2,3-双加氧酶 1 的酶促和非酶促功能的化合物

Panfili Eleonora, Rezzi Sarah Jane, Adamo Annalisa, Mazzoletti Daniele, Massarotti Alberto, Miggiano Riccardo, Fallarini Silvia, Ambrosino Sara, Coletti Alice, Molinaro Pasquale, Milella Michele, Paiella Salvatore, Macchiarulo Antonio, Ugel Stefano, Pirali Tracey, Pallotta Maria Teresa

Biological Evaluation of New Thienopyridinium and Thienopyrimidinium Derivatives as Human Choline Kinase Inhibitors

新型噻吩并吡啶和噻吩并嘧啶衍生物作为人胆碱激酶抑制剂的生物学评价

Luque-Navarro, Pilar María; Mariotto, Elena; Ballarotto, Marco; Rubbini, Gianluca; Aguilar-Troyano, Francisco José; Fasiolo, Alberto; Torretta, Archimede; Parisini, Emilio; Macchiarulo, Antonio; Laso, Alejandro; Marco, Carmen; Viola, Giampietro; Carrasco-Jimenez, María Paz; López-Cara, Luisa Carlota

Critical Assessment of a Structure-Based Screening Campaign for IDO1 Inhibitors: Tips and Pitfalls.

对基于结构的IDO1抑制剂筛选活动的关键评估:技巧和陷阱

Mammoli Andrea, Bianconi Elisa, Ruta Luana, Riccio Alessandra, Bigiotti Carlo, Souma Maria, Carotti Andrea, Rossini Sofia, Suvieri Chiara, Pallotta Maria Teresa, Grohmann Ursula, Camaioni Emidio, Macchiarulo Antonio

Environmentally Sustainable Achiral and Chiral Chromatographic Analysis of Amino Acids in Food Supplements

食品补充剂中氨基酸的非手性和手性色谱分析:环境可持续方法

Varfaj, Ina; Carotti, Andrea; Mangiapelo, Luciano; Cossignani, Lina; Taticchi, Agnese; Macchiarulo, Antonio; Ianni, Federica; Sardella, Roccaldo

Indoleamine 2,3-dioxygenase 1 (IDO1): an up-to-date overview of an eclectic immunoregulatory enzyme

吲哚胺2,3-双加氧酶1 (IDO1):一种多功能免疫调节酶的最新概述

Pallotta, Maria Teresa; Rossini, Sofia; Suvieri, Chiara; Coletti, Alice; Orabona, Ciriana; Macchiarulo, Antonio; Volpi, Claudia; Grohmann, Ursula