Discovery of a Series of 3-Cinnoline Carboxamides as Orally Bioavailable, Highly Potent, and Selective ATM Inhibitors
发现一系列3-肉桂酸甲酰胺类化合物作为口服生物利用度高、高效且选择性强的ATM抑制剂
期刊:ACS Medicinal Chemistry Letters
影响因子:4
doi:10.1021/acsmedchemlett.8b00200
Barlaam, Bernard; Cadogan, Elaine; Campbell, Andrew; Colclough, Nicola; Dishington, Allan; Durant, Stephen; Goldberg, Kristin; Hassall, Lorraine A; Hughes, Gareth D; MacFaul, Philip A; McGuire, Thomas M; Pass, Martin; Patel, Anil; Pearson, Stuart; Petersen, Jens; Pike, Kurt G; Robb, Graeme; Stratton, Natalie; Xin, Guohong; Zhai, Baochang