日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Diminishing GSH-Adduct Formation of Tricyclic Diazepine-based Mutant IDH1 Inhibitors

降低三环二氮杂卓类突变型IDH1抑制剂的GSH加合物形成

Huang, Chunhui; Fischer, Christian; Machacek, Michelle R; Bogen, Stephane; Biftu, Tesfaye; Huang, Xianhai; Reutershan, Michael H; Otte, Ryan; Hong, Qingmei; Wu, Zhicai; Yu, Yang; Park, Min; Chen, Lei; Biju, Purakkattle; Knemeyer, Ian; Lu, Ping; Kochansky, Christopher J; Hicks, Michael Brendan; Liu, Yong; Helmy, Roy; Fradera, Xavier; Donofrio, Anthony; Close, Josh; Maddess, Matthew L; White, Catherine; Sloman, David L; Sciammetta, Nunzio; Lu, Jun; Gibeau, Craig; Simov, Vladimir; Zhang, Hongjun; Fuller, Peter; Witter, David

Allosteric Modulation of Protein Arginine Methyltransferase 5 (PRMT5)

蛋白质精氨酸甲基转移酶 5 (PRMT5) 的变构调节

Palte, Rachel L; Schneider, Sebastian E; Altman, Michael D; Hayes, Robert P; Kawamura, Shuhei; Lacey, Brian M; Mansueto, My Sam; Reutershan, Michael; Siliphaivanh, Phieng; Sondey, Christopher; Xu, Haiyan; Xu, Zangwei; Ye, Yingchun; Machacek, Michelle R

Identification of predictive genetic signatures of Cytarabine responsiveness using a 3D acute myeloid leukaemia model.

利用 3D 急性髓系白血病模型鉴定阿糖胞苷反应性的预测性遗传特征

Xu Haiyan, Muise Eric S, Javaid Sarah, Chen Lan, Cristescu Razvan, Mansueto My Sam, Follmer Nicole, Cho Jennifer, Kerr Kimberley, Altura Rachel, Machacek Michelle, Nicholson Benjamin, Addona George, Kariv Ilona, Chen Hongmin

Sequential Ru-Pd catalysis: a two-catalyst one-pot protocol for the synthesis of N- and O-heterocycles

顺序Ru-Pd催化:一种用于合成N-和O-杂环化合物的双催化剂一锅法方案

Trost, Barry M; Machacek, Michelle R; Faulk, Brian D