日期 影响因子
日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:
–

Structure-activity relationship study of mesyl and busyl phosphoramidate antisense oligonucleotides for unaided and PSMA-mediated uptake into prostate cancer cells

甲磺酰基和布西酰基磷酰胺酯反义寡核苷酸在前列腺癌细胞中自发摄取和PSMA介导摄取的构效关系研究

期刊:Frontiers in Chemistry
影响因子:4.2
doi:10.3389/fchem.2024.1342178
Sergeeva, O; Akhmetova, E; Dukova, S; Beloglazkina, E; Uspenskaya, A; Machulkin, A; Stetsenko, D; Zatsepin, T
细胞生物学
肿瘤
前列腺癌
肿瘤免疫
发表日期：2024
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Synthesis and Preclinical Evaluation of Urea-Based Prostate-Specific Membrane Antigen-Targeted Conjugates Labeled with (177)Lu

尿素基前列腺特异性膜抗原靶向缀合物（177Lu标记）的合成及临床前评价

期刊:ACS Pharmacology and Translational Science
影响因子:3.7
doi:10.1021/acsptsci.4c00070
Machulkin, Aleksei E; Petrov, Stanislav A; Bodenko, Vitalina; Larkina, Mariia S; Plotnikov, Evgenii; Yuldasheva, Feruza; Tretyakova, Maria; Bezverkhniaia, Ekaterina; Zyk, Nikolay Yu; Stasyuk, Elena; Zelchan, Roman; Majouga, Alexander G; Tolmachev, Vladimir; Orlova, Anna; Beloglazkina, Elena K; Yusubov, Mekhman S
发表日期：2024
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Synthesis, 123I-Radiolabeling Optimization, and Initial Preclinical Evaluation of Novel Urea-Based PSMA Inhibitors with a Tributylstannyl Prosthetic Group in Their Structures

结构中含有三丁基锡烷基辅基的新型尿素基 PSMA 抑制剂的合成、123I 放射性标记优化及初步临床前评估

期刊:International Journal of Molecular Sciences
影响因子:0.7
doi:10.3390/ijms241512206
Lutfi A Hasnowo, Maria S Larkina, Evgenii Plotnikov, Vitalina Bodenko, Feruza Yuldasheva, Elena Stasyuk, Stanislav A Petrov, Nikolai Y Zyk, Aleksei E Machulkin, Nikolai I Vorozhtsov, Elena K Beloglazkina, Valentine G Nenajdenko, Vladimir Tolmachev, Anna Orlova, Alexander G Majouga, Mekhman S Yusubov
发表日期：2023
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Synthesis of Prostate-Specific Membrane Antigen-Targeted Bimodal Conjugates of Cytotoxic Agents and Antiandrogens and Their Comparative Assessment with Monoconjugates

前列腺特异性膜抗原靶向细胞毒剂和抗雄激素双峰结合物的合成及其与单结合物的比较评估

期刊:International Journal of Molecular Sciences
影响因子:0.7
doi:10.3390/ijms241411327
Nikolai Y Zyk, Anastasiia S Garanina, Ekaterina A Plotnikova, Anton P Ber, Ekaterina A Nimenko, Natalia S Dashkova, Anastasiia A Uspenskaia, Radik R Shafikov, Dmitry A Skvortsov, Stanislav A Petrov, Andrey A Pankratov, Nikolai V Zyk, Alexander G Majouga, Elena K Beloglazkina, Aleksei E Machulkin
细胞生物学
其它细胞
发表日期：2023
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Synthesis and Preclinical Evaluation of Small-Molecule Prostate-Specific Membrane Antigen-Targeted Abiraterone Conjugate

小分子前列腺特异性膜抗原靶向阿比特龙偶联物的合成及临床前评价

期刊:Molecules
影响因子:4.2
doi:10.3390/molecules27248795
Aleksei E Machulkin, Ekaterina A Nimenko, Nikolay U Zyk, Anastasiia A Uspenskaia, Galina B Smirnova, Irina I Khan, Vadim S Pokrovsky, Alexander N Vaneev, Roman V Timoshenko, Vugara V Mamed-Nabizade, Maria V Zavertkina, Alexander Erofeev, Petr Gorelkin, Alexander G Majouga, Nikolay V Zyk, Elena S Kha
信号转导
发表日期：2022
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Pharmacokinetic Properties of 68Ga-labelled Folic Acid Conjugates: Improvement Using HEHE Tag

68Ga 标记叶酸结合物的药代动力学特性：使用 HEHE 标签进行改进

期刊:Molecules
影响因子:4.2
doi:10.3390/molecules25112712
Anton Larenkov, Marat Rakhimov, Kristina Lunyova, Olga Klementyeva, Alesya Maruk, Aleksei Machulkin
发表日期：2020
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