日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Nintedanib Lacks Efficacy in a Spirometry-Confirmed and Bleomycin-Induced Mouse Model of Idiopathic Pulmonary Fibrosis.

尼达尼布在肺功能测定证实和博来霉素诱导的特发性肺纤维化小鼠模型中缺乏疗效。

Bousamaki Jamal, Maciag Grzegorz, Petersen Asbjørn Graver, Korntner Stefanie H, Jansen Stine Marie, Pors Susanne E, Mamsen Linn Salto, Rasmussen Silas A, Salinas Casper Gravesen, Kruse Louise Humle, Feigh Michael, Simonsen Ulf, Hansen Henrik H

Enzymes in secondary pharmacology screening panels: is there room for improvement?

二级药理学筛选组合中的酶:还有改进的空间吗?

Maciag, Monika; Karamyan, Vardan T

Discovery of BBO-8520, a First-In-Class Direct and Covalent Dual Inhibitor of GTP-Bound (ON) and GDP-Bound (OFF) KRASG12C.

发现 BBO-8520,一种首创的直接共价双重抑制剂,可抑制 GTP 结合 (ON) 和 GDP 结合 (OFF) 的 KRASG12C

Maciag Anna E, Stice James P, Wang Bin, Sharma Alok K, Chan Albert H, Lin Ken, Singh Devansh, Dyba Marcin, Yang Yue, Setoodeh Saman, Smith Brian P, Ju Jin Hyun, Jeknic Stevan, Rabara Dana, Zhang Zuhui, Larsen Erik K, Esposito Dominic, Denson John-Paul, Ranieri Michela, Meynardie Mary, Mehdizadeh Sadaf, Alexander Patrick A, Abreu Blanco Maria, Turner David M, Xu Rui, Lightstone Felice C, Wong Kwok-Kin, Stephen Andrew G, Wang Keshi, Simanshu Dhirendra K, Sinkevicius Kerstin W, Nissley Dwight V, Wallace Eli, McCormick Frank, Beltran Pedro J

Blocking C-terminal processing of KRAS4b via a direct covalent attack on the CaaX-box cysteine.

通过对 CaaX 盒半胱氨酸进行直接共价攻击,阻断 KRAS4b 的 C 端加工

Maciag Anna E, Yang Yue, Sharma Alok K, Turner David M, DeHart Caroline J, Abdelkarim Hazem, Fan Lixin, Smith Brian P, Kumari Vandana, Dyba Marcin, Rigby Megan, Castillo Badillo Jean A, Adams Lauren, Fornelli Luca, Fox Stephen, Brafman Alla, Turbyville Thomas, Gillette William, Messing Simon, Agamasu Constance, Wolfe Andrew L, Gysin Stephan, Chan Albert H, Simanshu Dhirendra K, Esposito Dominic, Chertov Oleg, Stephen Andrew G, Arkin Michelle, Renslo Adam, Kelleher Neil L, Gaponenko Vadim, Lightstone Felice C, Nissley Dwight V, McCormick Frank

The Missing Enzymes: A Call to Update Pharmacological Profiling Practices for Better Drug Safety Assessment

缺失的酶:呼吁更新药理学分析方法,以更好地评估药物安全性

Maciag, Monika; Karamyan, Vardan T

Microbial Enhancement of Plant Tolerance to Waterlogging: Mechanisms and Interplay with Biological Control of Pathogens

微生物增强植物耐涝性:机制及其与病原体生物防治的相互作用

Maciag, Tomasz; Krzyżanowska, Dorota M

Photocatalytic Activity of Thin Layers Obtained via Electrodeposition and Annealing of Nanostructured WFeZn and WFeCu Alloys

通过电沉积和退火法制备的纳米结构WFeZn和WFeCu合金薄层的光催化活性

Ratajczyk, Tomasz; Miecznikowski, Krzysztof; Majewski, Pawel; Maciag, Rafal; Donten, Mikolaj

The Genetic and Epigenetic Arms of Human Ageing and Longevity

人类衰老和长寿的遗传和表观遗传机制

Ciaglia, Elena; Montella, Francesco; Lopardo, Valentina; Basile, Cristina; Esposito, Roberta Maria; Maglio, Clara; Longo, Roberta; Maciag, Anna; Puca, Annibale Alessandro

In vivo evidence supports the effectiveness of the longevity-associated protein LAV-BPIFB4 in reducing adipose tissue-derived mediators of systemic inflammation to prevent vascular insult and atheromatous change

体内实验证据支持长寿相关蛋白LAV-BPIFB4能够有效减少脂肪组织来源的全身炎症介质,从而预防血管损伤和动脉粥样硬化。

Elena Ciaglia ,Valentina Lopardo ,Francesco Montella ,Roberta Maria Esposito ,Antonio Damato ,Angela Carmelita Abate ,Anna Maciag ,Carmine Vecchione ,Albino Carrizzo ,Annibale Alessandro Puca

NMR (1)H, (13)C, and (15)N resonance assignments of the oncogenic Q61R variant of human NRAS in the active, GTP-bound conformation

人类 NRAS 致癌 Q61R 变体在活性 GTP 结合构象下的 NMR (1)H、(13)C 和 (15)N 共振归属

Sharma, Alok K; Tonelli, Marco; Dyba, Marcin; Gillette, William K; Esposito, Dominic; Nissley, Dwight V; McCormick, Frank; Maciag, Anna E