日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Targeting Mediator Kinase Cyclin-Dependent Kinases 8/19 Potentiates Chemotherapeutic Responses, Reverses Tumor Growth, and Prolongs Survival from Ovarian Clear Cell Carcinoma.

靶向介导激酶细胞周期蛋白依赖性激酶 8/19 可增强化疗反应,逆转肿瘤生长,延长卵巢透明细胞癌患者的生存期

Barton Wade C, Kumari Asha, Mack Zachary T, Schools Gary P, Quintero Liz Macias, Choi Alex Seok, Rangavajhula Karthik, Arend Rebecca C, Broude Eugenia V, Mythreye Karthikeyan

Mediator kinase inhibition reverses castration resistance of advanced prostate cancer

介质激酶抑制剂可逆转晚期前列腺癌的去势抵抗性

Li, Jing; Hilimire, Thomas A; Liu, Yueying; Wang, Lili; Liang, Jiaxin; Gyorffy, Balazs; Sikirzhytski, Vitali; Ji, Hao; Zhang, Li; Cheng, Chen; Ding, Xiaokai; Kerr, Kendall R; Dowling, Charles E; Chumanevich, Alexander A; Mack, Zachary T; Schools, Gary P; Lim, Chang-Uk; Ellis, Leigh; Zi, Xiaolin; Porter, Donald C; Broude, Eugenia V; McInnes, Campbell; Wilding, George; Lilly, Michael B; Roninson, Igor B; Chen, Mengqian

Mediator kinase inhibitors suppress triple-negative breast cancer growth and extend tumor suppression by mTOR and AKT inhibitors

介导激酶抑制剂可抑制三阴性乳腺癌的生长,并延长mTOR和AKT抑制剂的肿瘤抑制作用。

Ding, Xiaokai; Liang, Jiaxin; Sharko, Amanda C; Hilimire, Thomas A; Li, Jing; Loskutov, Jürgen; Mack, Zachary T; Ji, Hao; Schools, Gary P; Cai, Chao; Pugacheva, Elena N; Chen, Mengqian; Roninson, Igor B; Broude, Eugenia V

Inhibition of CDK8/19 Mediator kinase potentiates HER2-targeting drugs and bypasses resistance to these agents in vitro and in vivo

抑制 CDK8/19 介导激酶可增强 HER2 靶向药物的疗效,并在体外和体内克服对这些药物的耐药性。

Ding, Xiaokai; Sharko, Amanda C; McDermott, Martina S J; Schools, Gary P; Chumanevich, Alexander; Ji, Hao; Li, Jing; Zhang, Li; Mack, Zachary T; Sikirzhytski, Vitali; Shtutman, Michael; Ivers, Laura; O'Donovan, Norma; Crown, John; Győrffy, Balázs; Chen, Mengqian; Roninson, Igor B; Broude, Eugenia V

Identifying Cancers Impacted by CDK8/19

识别受 CDK8/19 影响的癌症

Roninson, Igor B; Győrffy, Balázs; Mack, Zachary T; Shtil, Alexander A; Shtutman, Michael S; Chen, Mengqian; Broude, Eugenia V