Development of BET Inhibitors as Potential Treatments for Cancer: Optimization of Pharmacokinetic Properties
BET抑制剂作为潜在癌症治疗药物的开发:药代动力学特性的优化
期刊:ACS Medicinal Chemistry Letters
影响因子:4
doi:10.1021/acsmedchemlett.2c00219
Hill, Matthew D; Fang, Haiquan; Norris, Derek; Delucca, George V; Huang, Hong; DeBenedetto, Mikkel; Quesnelle, Claude; Schmitz, William D; Tokarski, John S; Sheriff, Steven; Yan, Chunhong; Fanslau, Caroline; Haarhoff, Zuzana; Huang, Christine; Kramer, Melissa; Madari, Shilpa; Menard, Krista; Monereau, Laura; Morrison, John; Raghavan, Nirmala; Shields, Eric E; Simmermacher-Mayer, Jean; Sinz, Michael; Tye, Ching Kim; Westhouse, Richard; Xie, Chunshan; Zhang, Haiying; Zhang, Lisa; Zvyaga, Tatyana; Lee, Francis; Gavai, Ashvinikumar V; Degnan, Andrew P