日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Combined treatment with CDK4/6, CDK2, and CXCR1/2 inhibitors effectively halts the growth of BRAF wild-type melanoma tumors.

CDK4/6、CDK2 和 CXCR1/2 抑制剂联合治疗可有效阻止 BRAF 野生型黑色素瘤肿瘤的生长

Yang Jinming, Luo Weifeng, Ward Patricia, Chen Sheau-Chiann, Zebala John, Maeda Dean, Yan Chi, Richmond Ann

Tumor-induced endothelial RhoA activation mediates tumor cell transendothelial migration and metastasis

肿瘤诱导的内皮细胞RhoA激活介导肿瘤细胞跨内皮迁移和转移

Sajib, Md Sanaullah; Zahra, Fatema Tuz; Lamprou, Margarita; Akwii, Racheal Grace; Park, Jee Hyun; Osorio, Manuel; Tullar, Paul; Doci, Colleen L; Zhang, Chonghe; Huveneers, Stephan; Van Buul, Jaap D; Wang, Ming-Hai; Markiewski, Maciej M; Srivastava, Sanjay K; Zheng, Yi; Gutkind, J Silvio; Hu, Junhao; Bickel, Ulrich; Maeda, Dean Y; Zebala, John A; Lionakis, Michail S; Trasti, Scott; Mikelis, Constantinos M

Regression and Eradication of Triple-Negative Breast Carcinoma in 4T1 Mouse Model by Combination Immunotherapies

联合免疫疗法在4T1小鼠模型中逆转和根除三阴性乳腺癌

Nahar, Saifun; Huang, Yue; Nagy, Bethany A; Zebala, John A; Maeda, Dean Y; Rudloff, Udo; Oppenheim, Joost J; Yang, De

Inhibiting myeloid-derived suppressor cell trafficking enhances T cell immunotherapy

抑制髓系来源抑制细胞的迁移可增强T细胞免疫疗法

Sun, Lillian; Clavijo, Paul E; Robbins, Yvette; Patel, Priya; Friedman, Jay; Greene, Sarah; Das, Rita; Silvin, Chris; Van Waes, Carter; Horn, Lucas A; Schlom, Jeffrey; Palena, Claudia; Maeda, Dean; Zebala, John; Allen, Clint T

Neutrophil content predicts lymphocyte depletion and anti-PD1 treatment failure in NSCLC

中性粒细胞含量可预测非小细胞肺癌中的淋巴细胞耗竭和抗PD-1治疗失败

Kargl, Julia; Zhu, Xiaodong; Zhang, Huajia; Yang, Grace H Y; Friesen, Travis J; Shipley, Melissa; Maeda, Dean Y; Zebala, John A; McKay-Fleisch, Jill; Meredith, Gavin; Mashadi-Hossein, Afshin; Baik, Christina; Pierce, Robert H; Redman, Mary W; Thompson, Jeffrey C; Albelda, Steven M; Bolouri, Hamid; Houghton, A McGarry

Desmetramadol Is Identified as a G-Protein Biased µ Opioid Receptor Agonist

去甲曲马多被鉴定为一种G蛋白偏向性μ阿片受体激动剂

Zebala, John A; Schuler, Aaron D; Kahn, Stuart J; Maeda, Dean Y

Desmetramadol Has the Safety and Analgesic Profile of Tramadol Without Its Metabolic Liabilities: Consecutive Randomized, Double-Blind, Placebo- and Active Comparator-Controlled Trials

去甲曲马多具有曲马多的安全性和镇痛效果,且无其代谢副作用:连续随机、双盲、安慰剂和活性对照试验

Zebala, John A; Searle, Shawn L; Webster, Lynn R; Johnson, Matt S; Schuler, Aaron D; Maeda, Dean Y; Kahn, Stuart J

Boronic acid-containing CXCR1/2 antagonists: Optimization of metabolic stability, in vivo evaluation, and a proposed receptor binding model

含硼酸的CXCR1/2拮抗剂:代谢稳定性优化、体内评价及受体结合模型

Maeda, Dean Y; Peck, Angela M; Schuler, Aaron D; Quinn, Mark T; Kirpotina, Liliya N; Wicomb, Winston N; Auten, Richard L; Gundla, Rambabu; Zebala, John A

Boronic acid-containing aminopyridine- and aminopyrimidinecarboxamide CXCR1/2 antagonists: Optimization of aqueous solubility and oral bioavailability

含硼酸的氨基吡啶和氨基嘧啶甲酰胺类CXCR1/2拮抗剂:水溶性和口服生物利用度的优化

Schuler, Aaron D; Engles, Courtney A; Maeda, Dean Y; Quinn, Mark T; Kirpotina, Liliya N; Wicomb, Winston N; Mason, S Nicholas; Auten, Richard L; Zebala, John A

Intestinal transport of aminopterin enantiomers in dogs and humans with psoriasis is stereoselective: evidence for a mechanism involving the proton-coupled folate transporter

在患有银屑病的犬和人体内,氨基蝶呤对映体的肠道转运具有立体选择性:质子偶联叶酸转运蛋白参与其中的机制的证据

Menter, Alan; Thrash, Breck; Cherian, Christina; Matherly, Larry H; Wang, Lei; Gangjee, Aleem; Morgan, Joel R; Maeda, Dean Y; Schuler, Aaron D; Kahn, Stuart J; Zebala, John A