Selective inhibition of mutant isocitrate dehydrogenase 1 (IDH1) via disruption of a metal binding network by an allosteric small molecule
通过变构小分子破坏金属结合网络选择性抑制突变异柠檬酸脱氢酶 1 (IDH1)
期刊:Journal of Biological Chemistry
影响因子:4
doi:10.1074/jbc.M114.608497
Gejing Deng, Junqing Shen, Ming Yin, Jessica McManus, Magali Mathieu, Patricia Gee, Timothy He, Chaomei Shi, Olivier Bedel, Larry R McLean, Frank Le-Strat, Ying Zhang, Jean-Pierre Marquette, Qiang Gao, Bailin Zhang, Alexey Rak, Dietmar Hoffmann, Eamonn Rooney, Aurelie Vassort, Walter Englaro, Yi Li,