日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Discovery of the DNA-PKcs inhibitor DA-143 which exhibits enhanced solubility relative to NU7441

发现 DNA-PKcs 抑制剂 DA-143,其溶解度较 NU7441 有所提高。

Zachary J Waldrip # ,Baku Acharya # ,Daniel Armstrong ,Maha Hanafi ,Randall R Rainwater ,Sharon Amole ,Madeline Fulmer ,Ana Clara Azevedo-Pouly ,Alaina Burns ,Lyle Burdine ,Brendan Frett ,Marie Schluterman Burdine

Discovery of a Napabucasin PROTAC as an Effective Degrader of the E3 Ligase ZFP91

发现 Napabucasin PROTAC 是 E3 连接酶 ZFP91 的有效降解剂

Maha Hanafi, Xinde Chen, Nouri Neamati