日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

A Novel NAMPT Inhibitor-Based Antibody-Drug Conjugate Payload Class for Cancer Therapy

一种新型的基于NAMPT抑制剂的抗体-药物偶联物有效载荷用于癌症治疗

Böhnke, Niels; Berger, Markus; Griebenow, Nils; Rottmann, Antje; Erkelenz, Michael; Hammer, Stefanie; Berndt, Sandra; Günther, Judith; Wengner, Antje M; Stelte-Ludwig, Beatrix; Mahlert, Christoph; Greven, Simone; Dietz, Lisa; Jörißen, Hannah; Barak, Naomi; Bömer, Ulf; Hillig, Roman C; Eberspaecher, Uwe; Weiske, Jörg; Giese, Anja; Mumberg, Dominik; Nising, Carl Friedrich; Weinmann, Hilmar; Sommer, Anette

IL3RA-Targeting Antibody-Drug Conjugate BAY-943 with a Kinesin Spindle Protein Inhibitor Payload Shows Efficacy in Preclinical Models of Hematologic Malignancies

靶向IL3RA的抗体药物偶联物BAY-943,携带驱动蛋白纺锤体蛋白抑制剂有效载荷,在血液系统恶性肿瘤的临床前模型中显示出疗效。

Kirchhoff, Dennis; Stelte-Ludwig, Beatrix; Lerchen, Hans-Georg; Wengner, Antje Margret; Ahsen, Oliver von; Buchmann, Pascale; Märsch, Stephan; Mahlert, Christoph; Greven, Simone; Dietz, Lisa; Erkelenz, Michael; Zierz, Ruprecht; Johanssen, Sandra; Mumberg, Dominik; Sommer, Anette

Implications of being born late in the active season for growth, fattening, torpor use, winter survival and fecundity

在活跃季节末期出生对生长、增肥、冬眠利用、冬季生存和繁殖力的影响

Mahlert, Britta; Gerritsmann, Hanno; Stalder, Gabrielle; Ruf, Thomas; Zahariev, Alexandre; Blanc, Stéphane; Giroud, Sylvain

The iterative gramicidin s thioesterase catalyzes peptide ligation and cyclization

迭代短杆菌肽硫酯酶催化肽连接和环化

Katharina M Hoyer, Christoph Mahlert, Mohamed A Marahiel