日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

A synergistic interaction between PRMT5 and LSD1 inhibitors in AML.

PRMT5 和 LSD1 抑制剂在急性髓系白血病中存在协同作用。

Param Nesteene Joy, Arceci Elisa, Fiorentino Francesco, Pignata Luca, Torre Denis, Gutiérrez-Trejo Nayeli, Fong Jia Yi, Goy Pierre-Alexis, Han Brenda Y, Lambona Chiara, Di Bello Elisabetta, Castiello Carola, Barone Marco, Schwarz Megan, Arrowsmith Cheryl, Ito Koichi, Scherle Peggy, Wee Dave Keng Boon, Ndoye Steven, Tabaglio Tommaso, Jeyasekharan Anand D, Lakshmanan Manikandan, Cirilli Roberto, Habisch Hansjörg, Madl Tobias, Mattevi Andrea, Valente Sergio, Mai Antonello, Guccione Ernesto

Dynamic epigenetic regulation of BCLAF1 splicing in acute myeloid leukemia

急性髓系白血病中BCLAF1剪接的动态表观遗传调控

Sgueglia, Giulia; Massaro, Crescenzo; Muro, Annamaria; Lettiero, Ida; D'Agostino, Erika; Favale, Gregorio; Simonelli, Nicla; Del Gaudio, Nunzio; Carafa, Vincenzo; De Marchi, Tommaso; Rotili, Dante; Valente, Sergio; Mai, Antonello; Sbardella, Gianluca; De Simone, Mariacarla; Altucci, Lucia; Dell'Aversana, Carmela

Tumor microenvironment-activated ferritin nanovector enables enhanced tumor delivery of KRAS(G12C) inhibitors and degraders

肿瘤微环境激活的铁蛋白纳米载体可增强KRAS(G12C)抑制剂和降解剂的肿瘤递送。

Abbinantefina, Annalisa Pia; Tito, Claudia; Masciarelli, Silvia; Tisci, Giada; Sortoluzzi, Siria; Ceci, Pierpaolo; Falvo, Elisabetta; Exertier, Cécile; Troilo, Francesca; Petrozza, Vincenzo; Mai, Antonello; Rotili, Dante; Fazi, Francesco; Colotti, Gianni

Combined computational and classical medicinal chemistry procedure to disclose novel pyrrole-based compounds as potential antituberculosis agents

结合计算和经典药物化学方法,发现新型吡咯类化合物作为潜在的抗结核药物。

Ragno, Rino; Zwergel, Clemens; Valente, Sergio; Astolfi, Roberta; Lambona, Chiara; Proia, Eleonora; Giuliani, Lidia; Franzblau, Scott G; Fioravanti, Rossella; Mai, Antonello

Structural snapshots of Pseudomonas aeruginosa LptB(2)FG and LptB(2)FGC reveal insights into lipopolysaccharide recognition and transport.

铜绿假单胞菌 LptB(2)FG 和 LptB(2)FGC 的结构快照揭示了脂多糖识别和运输的见解。

Fiorentino Francesco, Cervoni Matteo, Wang Yi, Urner Leonhard H, Sauer Joshua B, Tran Anh, Corey Robin A, Rotili Dante, Mai Antonello, Stansfeld Phillip J, Imperi Francesco, Yu Edward W, Su Chih-Chia, Robinson Carol V, Bolla Jani R

Activation and inhibition of sirtuins: From bench to bedside

sirtuins 的激活和抑制:从实验室到临床

Fiorentino, Francesco; Fabbrizi, Emanuele; Mai, Antonello; Rotili, Dante

Long noncoding RNA H19 promotes the acquisition of a mesenchymal-like invasive phenotype in mesothelial primary cells through an HDAC1-mediated WT1/Sp1 switch.

长链非编码 RNA H19 通过 HDAC1 介导的 WT1/Sp1 转换促进间皮原代细胞获得间充质样侵袭表型

Bontempi Giulio, Michetti Federica, Terri Michela, Battistelli Cecilia, Conigliaro Alice, Garbo Sabrina, Montaldo Claudia, Valente Sergio, Zwergel Clemens, Mai Antonello, Nahavandi Araghi Azadeh, Domenici Alessandro, Menè Paolo, Tripodi Marco, Strippoli Raffaele

A Xanthine Derivative With Novel Heat Shock Protein 90-Alpha Inhibitory and Senolytic Properties

一种具有新型热休克蛋白90-α抑制和衰老细胞清除特性的黄嘌呤衍生物

Atlante, Sandra; Cis, Luca; Pirolli, Davide; Gottardi Zamperla, Michela; Barbi, Veronica; Mai, Antonello; Zwergel, Clemens; Marcozzi, Serena; Giuliani, Maria Elisa; Bigossi, Giorgia; Lai, Giovanni; Orlando, Fiorenza; Giacconi, Robertina; Lattanzio, Fabrizia; Matacchione, Giulia; Giordani, Chiara; Bracci, Massimo; Olivieri, Fabiola; Boschi, Federico; Tabarelli De Fatis, Paola; Ivaldi, Giovanni Battista; Malavolta, Marco; Farsetti, Antonella; De Rosa, Maria Cristina; Gaetano, Carlo

Discovery of First-in-Class Carbonic Anhydrase/Histone Deacetylase Dual Inhibitors with Antiproliferative Activity in Cancer Cells

发现具有抗癌细胞增殖活性的首创碳酸酐酶/组蛋白去乙酰化酶双重抑制剂

Bozdag, Murat; Mroweh, Nabil; Raucci, Alessia; Angeli, Andrea; Peppicelli, Silvia; Biagioni, Alessio; Calorini, Lido; Trisciuoglio, Daniela; Ragno, Rino; Astolfi, Roberta; Giuliani, Lidia; Zwergel, Clemens; Valente, Sergio; Andreucci, Elena; Carta, Fabrizio; Mai, Antonello; Supuran, Claudiu T

Advancements in Hydrazide-Based HDAC Inhibitors: A Review of Recent Developments and Therapeutic Potential

基于酰肼的HDAC抑制剂的研究进展:近期进展及治疗潜力综述

Raucci, Alessia; Zwergel, Clemens; Valente, Sergio; Mai, Antonello