Sulfinyl Aziridines as Stereoselective Covalent Destabilizing Degraders of the Oncogenic Transcription Factor MYC.
亚磺酰基氮丙啶作为致癌转录因子MYC的立体选择性共价去稳定化降解剂
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doi:10.1101/2025.02.24.639755
Rosen Hannah T, Li Kelvin, Li Erin L, Currier Brynne, Brittain Scott M, Garcia Francisco J, Beard Diana C, Haenni-Holzinger Sandra, Dovala Dustin, McKenna Jeffrey M, Schirle Markus, Maimone Thomas J, Nomura Daniel K