日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

The Intricate Nonribosomal Assembly of a Potent Antifungal Lipopeptide from the Burkholderia cepacia Complex

伯克霍尔德氏菌复合体中一种强效抗真菌脂肽的复杂非核糖体组装

Zhong, Lei; Mühlenweg, Agnes; Hong, Dou; Yammine, Sarah; Poch, Annette; Xu, Dingchang; Kirimlioglu, Yasemin; Großgloß, Lisa; Boulanger, Malo; Graeger, Franziska; Seidel, Maria; Gemander, Manuel; Walther, Grit; Kemper, Sebastian; Dang, Tam; Royer, Monique; Mainz, Andi; Cociancich, Stéphane; Süssmuth, Roderich D

Synthesis of Derivatives of the Antibiotic Albicidin: The N-Terminal Fragment as Key to Control Potency and Resistance Mediated by the Binding Protein AlbA

抗生素白菌素衍生物的合成:N端片段是控制其效力和耐药性的关键,而耐药性是由结合蛋白AlbA介导的。

Kulike-Koczula, Marcel; Hommernick, Kay; Ghimire, Leela B; Kosol, Simone; Zborovsky, Lieby; Seidel, Maria; Sattler, Nicole; Mainz, Andi; Weston, John B; Ghilarov, Dmitry; Süssmuth, Roderich D

Paenilamicins are context-specific translocation inhibitors of protein synthesis.

帕尼拉霉素是具有特定环境的蛋白质合成转位抑制剂

Koller Timm O, Berger Max J, Morici Martino, Paternoga Helge, Bulatov Timur, Di Stasi Adriana, Dang Tam, Mainz Andi, Raulf Karoline, Crowe-McAuliffe Caillan, Scocchi Marco, Mardirossian Mario, Beckert Bertrand, Vázquez-Laslop Nora, Mankin Alexander S, Süssmuth Roderich D, Wilson Daniel N

Paenilamicins from the honey bee pathogen Paenibacillus larvae are context-specific translocation inhibitors of protein synthesis

来自蜜蜂病原体幼虫芽孢杆菌(Paenibacillus larvae)的类芽孢杆菌素是蛋白质合成的特异性转位抑制剂。

Koller, Timm O; Berger, Max J; Morici, Martino; Paternoga, Helge; Bulatov, Timur; Di Stasi, Adriana; Dang, Tam; Mainz, Andi; Raulf, Karoline; Crowe-McAuliffe, Caillan; Scocchi, Marco; Mardirossian, Mario; Beckert, Bertrand; Vázquez-Laslop, Nora; Mankin, Alexander; Süssmuth, Roderich D; Wilson, Daniel N

Molecular mechanism of topoisomerase poisoning by the peptide antibiotic albicidin

肽类抗生素白菌素对拓扑异构酶的毒害分子机制

Michalczyk, Elizabeth; Hommernick, Kay; Behroz, Iraj; Kulike, Marcel; Pakosz-Stępień, Zuzanna; Mazurek, Lukasz; Seidel, Maria; Kunert, Maria; Santos, Karine; von Moeller, Holger; Loll, Bernhard; Weston, John B; Mainz, Andi; Heddle, Jonathan G; Süssmuth, Roderich D; Ghilarov, Dmitry

Transcription activation by the resistance protein AlbA as a tool to evaluate derivatives of the antibiotic albicidin

利用抗性蛋白AlbA的转录激活作用来评价抗生素白菌素衍生物

Kosol, Simone; Rostock, Lida; Barsig, Jonas; Tabarelli, Theresa; Hommernick, Kay; Kulike, Marcel; Eulberg, Tobias; Seidel, Maria; Behroz, Iraj; Kleebauer, Leonardo; Grätz, Stefan; Mainz, Andi; Süssmuth, Roderich D

Acetylenic Replacement of Albicidin's Methacrylamide Residue Circumvents Detrimental E/Z Photoisomerization and Preserves Antibacterial Activity

用乙炔基取代白菌素中的甲基丙烯酰胺残基可避免有害的E/Z光异构化并保持其抗菌活性。

Behroz, Iraj; Kleebauer, Leonardo; Hommernick, Kay; Seidel, Maria; Grätz, Stefan; Mainz, Andi; Weston, John B; Süssmuth, Roderich D

An Amphipathic Alpha-Helix Guides Maturation of the Ribosomally-Synthesized Lipolanthines

两亲性α螺旋引导核糖体合成的脂嘌呤的成熟

Wiebach, Vincent; Mainz, Andi; Schnegotzki, Romina; Siegert, Mary-Ann J; Hügelland, Manuela; Pliszka, Nicole; Süssmuth, Roderich D

Harnessing fungal nonribosomal cyclodepsipeptide synthetases for mechanistic insights and tailored engineering

利用真菌非核糖体环状缩肽合成酶进行机制研究和定制工程改造

Steiniger, Charlotte; Hoffmann, Sylvester; Mainz, Andi; Kaiser, Marcel; Voigt, Kerstin; Meyer, Vera; Süssmuth, Roderich D

Structural and mechanistic implications of metal binding in the small heat-shock protein αB-crystallin

金属结合在小热休克蛋白αB-晶状体蛋白中的结构和机制意义

Mainz, Andi; Bardiaux, Benjamin; Kuppler, Frank; Multhaup, Gerd; Felli, Isabella C; Pierattelli, Roberta; Reif, Bernd